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2-(2,3-difluorophenoxymethyl)-4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,3-oxazole
(1R,5R)-3-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2,3-dimethoxy-N-methylbenzamide
4-{1-ethyl-5-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-1H-1,2,4-triazol-3-yl}benzamide
N-[3-(1H-imidazol-1-yl)propyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
4-methyl-5-{4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}pyrimidine
N5-(2-methoxyethyl)-N6-(3-methoxypropyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-(3,5-dimethoxyphenyl)-3-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}propanamide
3-(1-phenylethyl)-3H,4H-pyrido[2,3-d]pyrimidin-4-one
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(4-hydroxyphenyl)propan-1-one
8-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-methyl-1'-(4-methyl-1H-imidazole-5-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-[(5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-2-methoxyphenyl)methyl]-1H-1,2,4-triazole
N-methyl-N-[(5-methyl-1H-indol-3-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
(5S,9aS,9bS)-5-[(E)-2-(4-hydroxy-3-methoxyphenyl)ethenyl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(dimethylamino)-2-[2-(4-fluorophenyl)ethyl]-2,3-dihydropyridazin-3-one
N-butyl-1-(furan-2-ylmethyl)-5-(3-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(2R,4S)-1-(2-ethylbutanoyl)-4-hydroxypiperidine-2-carboxylic acid
5-{[(2,6-dimethoxyphenyl)methyl]amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
3-cyclopentyl-1-[1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
3-{3-[(benzyloxy)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4-methyl-1,2,5-oxadiazole
6-[(4-fluorophenyl)methoxy]-4-[3-(2-oxoimidazolidin-1-yl)benzoyl]-1-(propan-2-yl)-1,4-diazepan-2-one
2-(2-methoxyethyl)-8-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1,2,3,4-tetrahydroquinoline-8-carboxamide
3-[(3S,4R)-1-benzyl-4-(morpholin-4-yl)piperidin-3-yl]-N-[(2-chlorophenyl)methyl]propanamide
3-{2-[(4aS,8aR)-decahydroisoquinolin-2-yl]-2-oxoethyl}-1-cyclopropyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-methyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(2H-1,3-benzodioxol-5-yl)-1-(1-cyclohexanecarbonylpiperidin-4-yl)-5-fluoro-1H-1,3-benzodiazole
3-chloro-N-cyclopentyl-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
N-methyl-N-(2-methylpropyl)-3-{[2-(2-oxoimidazolidin-1-yl)ethyl]sulfamoyl}benzamide
methyl 3-(2,4-dimethylbenzamido)-6-{[methyl(thiophen-2-ylmethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
1-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
4-(2,6-dimethylpyridine-4-carbonyl)-4-azatricyclo[4.3.1.13,8]undecane
9-(5-fluoro-2-methylbenzenesulfonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
4-{[3-chloro-5-ethoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-one
methyl({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl})(quinoxalin-6-ylmethyl)amine
4-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-propylpyrrolidin-2-one
3-(3,4-difluorophenyl)-5-(2-methoxy-6-methylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(1-{2-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
7-{[3-(4-chlorophenoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1'-(4-fluoro-2-methylbenzoyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[2-(dimethylamino)ethyl]-5-[1-(4-methylpentanoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-1,3-thiazole-4-carboxamide