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N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-2-methoxy-N-(2-methoxyethyl)benzamide
5-(3,4-dimethylphenoxymethyl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
3-(2-fluorophenyl)-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazole-5-carboxamide
4-[4-(2-methoxyacetyl)-1,4-diazepane-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
(2R,3R)-3-[butyl(methyl)amino]-1'-(furan-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}(methyl)(pyridin-2-ylmethyl)amine
2-cyclopropyl-8-[(2,3-difluoro-4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(3,4-dimethoxyphenyl)methyl]-3-fluoro-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-2-yl]pyridine
2-(1-{1-[(1-benzyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-2-(2-oxopiperidin-1-yl)acetamide
1'-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-4-ol
1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
6-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-4-methyl-1H,2H,3H-pyrazolo[3,4-b]pyridin-3-one
methyl (2S)-2-{[1-(3-cyclopropaneamidophenyl)piperidin-4-yl]amino}-3-phenylpropanoate
2-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,3-thiazole-4-carboxamide
3-{2-[(2-methyl-6-propylpyrimidin-4-yl)amino]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(4-aminophenyl)-6-methyl-1,3-benzothiazol-2-amine
1-ethyl-3-(2-methylpropyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
N-[(3S,4R)-1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
N-tert-butyl-2-(2-methylquinazolin-4-yl)benzene-1-sulfonamide
4-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}thiomorpholine
N4,N4,5-trimethyl-N2-[(1-propyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
4-(4-chlorophenyl)-1-[2-(hydroxymethyl)piperidin-1-yl]butan-1-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(propan-2-yl)piperidine-3-carboxylate
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-yl]methanol
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-6-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-{3-methyl-1-oxo-1-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]butan-2-yl}acetamide
ethyl 5-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-methoxy-5-methylthiophene-2-carboxamide
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
2-[(E)-2-[3-(4H-1,2,4-triazol-4-yl)phenyl]ethenyl]pyridine
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-cycloheptyl-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
(2S,4S)-4-amino-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-methylpyrrolidine-2-carboxamide
5-[(2,6-difluorophenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}pyridine-2-carboxamide
8-fluoro-3-{imidazo[1,2-a]pyridin-2-ylmethyl}-3,4-dihydroquinazolin-4-one
3-methyl-1-[2-(morpholin-4-ylmethyl)phenyl]-3-[1-(thiophen-2-yl)ethyl]urea
N-(4-cyano-2-ethylphenyl)-3-{[3-(hydroxymethyl)morpholin-4-yl]methyl}benzamide
1-[(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-oxazol-5-yl)methyl]piperidin-4-ol
1-[(2-methoxyphenyl)methyl]-N-[2-(5-methylfuran-2-yl)ethyl]-6-oxopiperidine-3-carboxamide