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4-(2,3-dihydro-1-benzofuran-2-carbonyl)-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-(piperidin-1-yl)ethan-1-one
6-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrazine-2-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
N-methyl-N-[4-(morpholin-4-yl)butyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
N-butyl-N-[(2-methylphenyl)methyl]-1,1-dioxo-1λ6-thiane-4-carboxamide
3-(5-{3-[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]propyl}-1,2,4-oxadiazol-3-yl)pyridine
2-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
7-[(2,4-difluorophenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(oxolan-2-ylmethyl)-3-{[2-(1H-pyrazol-1-yl)ethyl]sulfamoyl}benzamide
3-(3-hydroxy-3-methylbutyl)-N-[2-methyl-1-(pyridin-2-yl)propyl]benzamide
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
1-cyclopropyl-N-methyl-6-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[methyl(pyridin-3-ylmethyl)amino]-1-[4-(naphthalen-2-yl)piperazin-1-yl]ethan-1-one
2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(2-phenylethyl)acetamide
N-cyclopropyl-3-(4-{[methyl(thian-4-yl)carbamoyl]amino}phenyl)propanamide
(2E)-1-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
4-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-1-ethyl-1H-pyrrole-2-carbonitrile
2-{[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]methyl}-1,3-benzoxazole
9-(cyclopropylmethyl)-4-[(5-ethylfuran-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(3,4-difluorophenyl)-2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
2-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-3,4,7-trimethyl-1H-indole
2-methyl-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)benzamide
1-[benzyl(methyl)amino]-3-(5-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
(3S,5S,9R)-5-{[(3-chlorophenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
methyl 4-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}benzoate
7-(2-methoxyethyl)-2-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
2-(2-{[1-(4-methylpyridin-2-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-amino-6-(4-chlorophenyl)-4-[2-(ethylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-4-(pyridin-4-yl)piperazine-1-carboxamide
(1R,5S,6R)-3-(5-carboxypyrimidin-4-yl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
(4aS,7aR)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[ethyl({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)amino]ethan-1-ol
3-(2-methoxy-5-methylbenzenesulfonyl)-3,9-diazaspiro[5.6]dodecan-10-one
(4aS,7aR)-1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-4-(1H-imidazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(3-aminopyrrolidine-1-carbonyl)-2-(3,5-dichlorophenyl)pyrimidin-4-ol
[(5-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
3-(3,4-dimethylphenyl)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,4-dimethyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]propanamide
6-methyl-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-2-oxo-1,2-dihydropyridine-4-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amine
N-methyl-N-[2-(oxan-2-yl)ethyl]-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetamide
2-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-2-yl}pyridine
4-methoxy-2-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidine
N-ethyl-3-fluoro-N-(oxan-2-ylmethyl)pyridine-4-carboxamide
1-(benzenesulfonyl)-N-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-4-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(propan-2-yl)pyrimidine-5-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide