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3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]piperidine-1-carboxamide
8-benzyl-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-phenylpyrrolidine-3-carboxylic acid
2-(2,5-dioxoimidazolidin-4-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]acetamide
5-phenyl-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1H-pyrrole-2-carboxamide
1-cyclopentyl-3-(2-methoxyphenyl)-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-1,2-dimethyl-1H-indol-5-ol
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
(1S,5R)-6-(4-ethyl-5-methylthiophene-3-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-ethyl-3-[(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)methyl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-(1,3-thiazol-2-ylmethyl)piperidin-2-yl]pyridine
ethyl 1-(3-phenylpropyl)-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-({5-[(3-ethoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
methyl 2-(azepane-1-sulfonyl)-6-(4-fluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{1-[1-(2-cyclopropylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[5-(pyridin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
4-(4-ethyl-2,3-dioxopiperazin-1-yl)-2,2-diphenylbutanenitrile
4-ethyl-5-[2-(4-methylpentyl)morpholine-4-carbonyl]-1,3-thiazol-2-amine
2-(3-fluorophenyl)-N-{[7-(quinolin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(thiophen-2-ylmethyl)benzamide
3-[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]-N-(1,3-thiazol-2-yl)propanamide
3-(1-methylpiperidin-2-yl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]propan-1-one
(2S,3R)-3-hydroxy-2-({5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazol-3-yl}formamido)butanamide
(3R,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-(thiophen-3-ylmethyl)pyrrolidin-3-amine
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[4-(methylsulfanyl)butan-2-yl]piperidine
1-[2-(3-chloro-4-hydroxyphenyl)acetyl]-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[2-(3-fluorophenyl)-2-hydroxyethyl]-2-(1-propylpiperidin-4-yl)acetamide
2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
1-(cyclohex-1-ene-1-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
4-(1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carbonyl)piperazine-1-carbaldehyde
4-fluoro-3-[2-(furan-2-yl)azepane-1-carbonyl]benzene-1-sulfonamide
5-methyl-1'-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
2-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}benzoic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(pyridin-3-ylmethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-[(4-chlorophenyl)methyl]-N-[5-(morpholin-4-yl)pentyl]-1,3-benzoxazole-5-carboxamide
4-(2,2-diphenylethyl)-4H-1,2,4-triazole
2-(4-fluorophenoxymethyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
(3R,4R)-3,4-dimethyl-1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-3-ol
4-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5-methyl-1,3-oxazole
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-(4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylphenyl)-1H-pyrrole
N-[(2R,3R)-2-ethoxy-1'-(1,3-thiazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
1-[(4-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(2-fluorophenyl)piperazine
1-{1-[(2-aminopyrimidin-5-yl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide