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N-(3-chloro-4-methoxyphenyl)-3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)propanamide
1-cyclopropanecarbonyl-4-{4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]phenoxy}piperidine
1-{1-[(4-fluoro-2-methoxyphenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
(3S,9aR)-8-(2,5-difluorobenzoyl)-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-7-(thiophene-2-sulfonamido)-1H-1,3-benzodiazole-5-carboxamide
(1R,5R)-3-[4-(methylsulfanyl)benzoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1-[1-(5-fluoro-1H-indole-2-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methyloxane-4-carboxamide
2-{1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-cycloheptanecarbonyl-3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
5-ethyl-N-[2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-(2-methoxyphenyl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
4-[4-(thiophen-3-ylmethyl)piperazin-1-yl]pyrimidine-5-carboxylic acid
4-[(dimethylamino)methyl]-1-[2-(methylamino)pyridine-3-carbonyl]azepan-4-ol
N-butyl-2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)acetamide
ethyl({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})[(1-methyl-1H-pyrazol-4-yl)methyl]amine
7-(2-methoxyethyl)-2-[3-(thiophen-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
5-methyl-1-(4-methylphenyl)-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazin-2-one
4-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)morpholine-2-carboxamide
1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-(2,2,2-trifluoroethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(4-methoxyphenyl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-amine
N-[(2-fluorophenyl)methyl]-1-methyl-5-[(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-methanesulfonyl-4-[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]piperidine
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})(propan-2-yl)amine
1-benzyl-4-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-1,4-diazepan-6-ol
1-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazole
2,3-dimethyl-6-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]quinoxaline
2-methoxy-1-[4-(2-phenylazetidine-1-carbonyl)piperidin-1-yl]ethan-1-one
3-(1H-1,2,3-benzotriazol-1-yl)-1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]propan-1-one
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
N-methyl-6-(piperidin-3-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
N-cyclopropyl-4-oxo-N-(3-phenylprop-2-yn-1-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-methyl-3-(2-phenylethyl)-8-[(4-phenylphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(propan-2-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1H-pyrazole-3-carboxamide
4-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
N-(1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
2-[3-(2-aminoethyl)piperidin-1-yl]-N-(2-ethylphenyl)-2-oxoacetamide
1-{2-[3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-yl}pyrrolidin-3-ol
3-(1,4-dioxan-2-ylmethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(5-chloropyridin-2-yl)-4-(1H-imidazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-ethyl-N-(thiolan-3-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-({2-[1-(7-methyl-1-benzofuran-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(1S,6R)-9-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
4-{1-[6-(4-methoxypiperidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
1-[7,8-dimethyl-2-(pyrimidin-5-yl)quinoline-4-carbonyl]-N,N-dimethylpiperidin-4-amine
(1s,4s)-4-{4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
ethyl 4-(cyclopropylmethyl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine-4-carboxylate
N-(3-cyclopentylpropyl)-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methylbenzamide
3-(2-methoxyethyl)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-3-carboxylic acid