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3-chloro-4-fluoro-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzothiophene-2-carboxamide
N-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)methanesulfonamide
2-[(2-hydroxyethoxy)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[(3R,4S)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
6-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-(4-methoxyphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]propanamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{[2-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidin-3-amine
2-(4-chlorophenyl)-1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
N-[(1-methylpiperidin-3-yl)methyl]-5-phenyl-N-(2-phenylethyl)-1,2-oxazole-4-carboxamide
methyl 4-[5-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
ethyl 3-[(3-methoxyphenyl)methyl]-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidine-3-carboxylate
6-(benzyloxy)-1-cyclohexyl-4-(2-methyl-1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
2-[3-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-ethylpiperidine
N-methyl-3-(5-methylfuran-2-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-2-(pyrrolidin-1-yl)pyrimidine
3-chloro-2-[4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-indole
{5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]furan-2-yl}methanol
1-ethyl-N-[phenyl(pyridin-4-yl)methyl]piperidine-4-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2,7-diazaspiro[4.5]decane-7-sulfonyl}-2,5-dihydro-1λ6-thiophene-1,1-dione
1-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]urea
N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyridine-4-carboxamide
N-[(2R,3R)-2-methoxy-1'-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
(2R,6S)-2,6-dimethyl-4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)morpholine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyrazine-2-carbonyl)piperidin-4-amine
methyl 1-{2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-4-carboxylate
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
5-chloro-2-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazine-1-carbonyl]-2,3-dihydro-1H-indole
N-(9H-fluoren-9-yl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-methyl-3-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}propanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(pyrrolidine-1-sulfonyl)piperidine
5-[2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
N-ethyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-(1-benzothiophene-2-sulfonyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
3-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N5-cyclopentyl-N6-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[(diethylamino)methyl]-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
4-cyclobutanecarbonyl-2-[(4-methoxyphenyl)methyl]morpholine
1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
4-benzyl-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-(2-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]pyridine-4-carboxamide
N-[3-(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)-4-chlorophenyl]acetamide
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})amine
1-[(2S)-2-amino-4-methylpentanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine