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(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(ethanesulfonyl)-decahydro-1,6-naphthyridin-2-one
ethyl 5-[(2,6-difluorophenyl)methyl]-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
({4-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]benzamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
5-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
(2R,4S)-1-(2,3-dimethyl-1H-indole-7-carbonyl)-4-hydroxypiperidine-2-carboxylic acid
5-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
5-(4-cyclohexylphenyl)-3-(1,2-oxazolidin-2-yl)-1,2,4-triazine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(2S)-1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}pyrrolidine-2-carboxamide
3-cyclopropyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1H-pyrazole-5-carboxamide
3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[2-(piperidin-1-yl)ethyl]propanamide
2-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-phenylbenzamide
5-ethyl-N-[3-(pyridin-3-yl)propyl]-1,3,4-oxadiazol-2-amine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethylbenzamide
1-(2-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
7-[2-(phenylamino)pyrimidine-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3R,4S)-4-[4-(1-benzothiophene-5-carbonyl)-1,4-diazepan-1-yl]oxolan-3-ol
3-fluoro-5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]benzonitrile
6-(4-ethyl-5-methylthiophene-3-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}benzamide
2-(2-ethyl-1H-imidazol-1-yl)-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}morpholine-2-carboxamide
3-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
4-(2H-1,3-benzodioxol-5-yl)-2-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
2-(3,5-difluoro-4-methoxyphenyl)-1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazole
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-(4-propanoylphenoxy)acetamide
(2S)-3-(1H-imidazol-4-yl)-2-[(5-propyl-1,2-oxazol-3-yl)formamido]propanamide
7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
5-methyl-1'-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 1-[2-(dimethylamino)ethyl]-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}piperidin-2-one
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(pyridin-4-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[4-(3-methyl-1H-pyrazol-4-yl)benzoyl]piperidine
N-methyl-4-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
(4aR,8aR)-1-(2,4-dimethoxybenzoyl)-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridine
N-(2,3-dihydro-1H-inden-1-yl)-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-{[(1-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
(1S,5R)-6-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-1,3-diazinane-2,4-dione
7-fluoro-4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methylquinoline
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(pyridin-4-ylsulfanyl)acetamide
N-cyclohexyl-N-methyl-3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine