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1-[2-(4-methylpentyl)morpholin-4-yl]-2-(pyridin-3-yl)ethan-1-one
N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
[(3-chloropyridin-4-yl)methyl]({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})methylamine
1-(5-chloro-2-methoxyphenyl)-3-(oxan-4-yl)-5-(1H-pyrazol-4-yl)-1H-1,2,4-triazole
1-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
6-{4-[1-(dimethylamino)ethyl]phenyl}-N,N-dimethylpyrazine-2-carboxamide
1-(2-methylphenyl)-4-{1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}piperazine
N-ethyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(2,4-difluorophenyl)methyl]piperidine-3-carboxamide
6-{1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
2-methyl-N-(1-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
4-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-(2-hydroxyethyl)piperazin-2-one
1-(2-ethoxyethyl)-5-[4-(2-hydroxyethyl)piperidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(3-methyl-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}-1H-1,2,4-triazol-1-yl)acetic acid
N-{[(1R,2S,5R)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl]methyl}-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(phenylsulfanyl)acetamide
2-(3-methoxyphenyl)-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
1-benzyl-8-(1H-indol-3-ylmethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(butylcarbamoyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
N-(1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
4-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}morpholine
2-(2-hydroxyethyl)-9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(cyclopentylamino)-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-{3-[2-(3-cyanophenyl)-1H-imidazol-1-yl]-4-fluorophenyl}methanesulfonamide
(3aS,6aR)-5-(cyclopropylmethyl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
1-methyl-9-(2-phenylquinazolin-4-yl)-1,4,9-triazaspiro[5.5]undecan-5-one
5-[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-methoxy-3-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrazine
2-ethyl-N-methyl-N-[(4-phenylphenyl)methyl]pyrimidine-5-carboxamide
2-(3-{4-[(2-cyanophenyl)methyl]piperazine-1-carbonyl}piperidin-1-yl)acetamide
7,7-dimethyl-2-(3-methylthiophen-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}cyclopentane-1,3-dicarboxamide
4-(3-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2,2-dimethylpropyl)morpholine
(1S,5R)-3-cyclobutanecarbonyl-6-(4-ethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-methyl-1H-indazol-3-yl)-3-[(2-methylpyrrolidin-1-yl)methyl]benzamide
1-(3-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-3-oxopropyl)-6-methyl-1,2-dihydropyridin-2-one
3-{2-[1-(pyridin-3-ylmethyl)piperidin-2-yl]ethyl}phenol
N-[(2R,3R)-1'-[(2,5-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
N-(2,4-difluorophenyl)-3-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}benzamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-3-yl]methanol
(3S,4S)-4-cyclopropyl-1-[3-(1H-pyrazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
2-[(cyclooctylamino)methyl]-4-(pyridin-2-yl)phenol
N-[(3S,5S)-5-{[2-(1H-imidazol-1-yl)ethyl]carbamoyl}-1-methylpyrrolidin-3-yl]morpholine-4-carboxamide
methyl 6-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}pyridine-2-carboxylate
3-cyano-N-{3-[(dimethylsulfamoyl)amino]phenyl}piperidine-1-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-(methylsulfanyl)benzamide
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-[4-(4-methoxybenzoyl)piperazin-1-yl]propan-1-one
2-methyl-1-[5-(pyrrolidine-1-carbonyl)furan-2-yl]-1H-1,3-benzodiazole-4-carboxylic acid