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N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-methyl-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
N-(2-methoxyethyl)-1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-{1H-pyrazolo[3,4-b]pyridin-1-ylmethyl}-1,3-oxazole
N-{[3-(methylsulfanyl)phenyl]methyl}-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
(5S)-5-[3-(2,2-diphenylethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
1-(oxolan-2-ylmethyl)-4-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperazine
2-(2,3-dihydro-1H-inden-1-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
5-methyl-3-[5-(2,3,4-trifluorobenzenesulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-cyclohexyl-N-(pyridin-4-ylmethyl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
3-(4-cyano-4-phenylpiperidine-1-carbonyl)piperidine-1-carboxamide
2-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
3-methoxy-1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidine
(2R,3S,6R)-5-(cyclopropanesulfonyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
3-methyl-7-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
4-(4-{[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenyl)but-3-yn-1-ol
2-methyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-(1-{[1-(2-methylpentyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-1-ol
2-{4-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-1-methylpiperazin-2-yl}ethan-1-ol
N'-(adamantan-1-yl)-N-ethyl-N-(oxolan-2-ylmethyl)propanediamide
(2R,3S,6R)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3aS,6aS)-2-(2,4-difluorobenzoyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-ethyl-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
2-cyclopropyl-9-[2-(4-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(1s,4s)-4-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclohexan-1-ol
3-fluoro-4-[4-(pyridin-4-yl)piperidin-1-yl]pyridine
9-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]methanesulfonamide
N-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-(morpholin-4-yl)azetidine-1-carboxamide
1-[(4-chlorophenyl)methyl]-N-[1-(2-methoxyphenyl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-1-benzyl-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-{5-[(2,4-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(2-hydroxyethyl)propanamide
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}butan-1-one
3-[1-(1-ethylpiperidin-3-yl)piperidin-3-yl]propan-1-ol
N-[1-(2,5-difluorophenyl)cyclopropyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
4-(furan-3-yl)-6-(trifluoromethyl)-1H-1,3-benzodiazole
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
3-{2-oxo-2-[2-(pyrrolidin-1-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-(6-cyclopropylpyrimidin-4-yl)-4-(furan-3-carbonyl)-1,4-diazepane
4-[5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine