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1-(propan-2-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
N-[2-(1,3-benzothiazol-2-yl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
methyl 3-[(3,5-dimethoxyphenyl)methyl]-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
N4-[1-(1,3-thiazol-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-ethyl-3-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(furan-2-yl)-4-phenyl-1H-imidazole
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
3-{1-[1-(4-methoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclobutan-1-amine
6-methyl-4-[4-(oxolan-2-ylmethyl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(3-methylfuran-2-carbonyl)piperidine
N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(piperidin-1-yl)ethyl]acetamide
N-(3-hydroxypropyl)-2-[5-oxo-3-phenyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
N-(oxolan-3-ylmethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-4-(1H-pyrazol-4-yl)butanamide
1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-[(3,4-dichlorophenyl)methyl]piperazine
1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
3-{thieno[2,3-d]pyrimidin-4-yl}-4H-chromen-4-one
6,7-dimethoxy-3-{[(2S)-2,4,5,5-tetramethylpiperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
6-butyl-2-{4-[(2-methylpyrrolidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-ethylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(1R,5R)-3-(dimethylsulfamoyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-(furan-2-ylmethyl)propanamide
N6-cyclopropyl-N4-methyl-N4-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidine-2,4,6-triamine
(2S)-2-amino-N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-3-(1H-imidazol-4-yl)propanamide
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{5-[1-(2,5-dimethoxyphenyl)-1H-imidazol-2-yl]furan-2-yl}methanol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N,N-dimethyl-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazine-1-sulfonamide
3-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-2H-chromen-2-one
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
N-[3,3-dimethyl-1-(pyrrolidin-1-yl)butan-2-yl]-3-(5-methyl-4H-1,2,4-triazol-3-yl)propanamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(4-fluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(oxolan-3-yl)benzamide
8-[(4-hydroxyphenyl)methyl]-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-fluorophenyl)methyl]acetamide
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-3-propoxypiperidine
5-benzenesulfonamido-N-[(2,5-difluorophenyl)methyl]-1-ethyl-2-methyl-1H-1,3-benzodiazole-7-carboxamide
4-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
8-[(5-acetylthiophen-3-yl)methyl]-2-benzyl-2,8-diazaspiro[4.5]decan-3-one
5-{[({3-[2-(4-cyclopropanecarbonylpiperazin-1-yl)ethoxy]phenyl}methyl)(methyl)amino]methyl}pyrrolidin-2-one
ethyl 1-[(4-{[(3,4-dimethoxyphenyl)methyl](methyl)amino}quinazolin-2-yl)methyl]piperidine-2-carboxylate
3-(1-methylpiperidin-2-yl)-1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]propan-1-one
N-{1-[1-(2-methoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2-methyl-N-(pyridin-4-ylmethyl)propanamide
1-[4-(4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
3-chloro-5-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine