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N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(methylsulfanyl)pyridine-3-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-{[(propan-2-yl)amino]methyl}piperidin-2-one
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]azetidin-3-ol
5-(3-methylphenyl)-4-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-2-(pyridin-4-yl)pyrimidine
3-hydroxy-3-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}-1-(2-phenylethyl)piperidin-2-one
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-5-methyl-1H-pyrazole-3-carboxamide
1,3,5-trimethyl-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-1H-pyrazole-4-sulfonamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-phenoxypropan-1-one
(3S,4S)-1-(1H-indole-2-carbonyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
1-[2-(dimethylamino)ethyl]-4-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
(3S,4R)-1-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-4-phenylpyrrolidine-3-carboxylic acid
2-amino-N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
[(1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]urea
1-cyclopentyl-4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-methyl-5-{[3-(2-phenylethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
2-[(3aR,6aR)-2-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-1,2,3,4-tetrahydroisoquinoline
3-{1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
N-[(2-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)spiro[2.2]pentane-1-carboxamide
methyl({5-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)(1,2-oxazol-5-ylmethyl)amine
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-(pyrrolidin-3-yl)benzamide
6-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carboxylic acid
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[(4-fluorophenyl)methyl]-N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
3-(4-methylpiperazine-1-carbonyl)-1-propyl-N-{[2-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)morpholine
4-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
N-[(3,4-dimethoxyphenyl)methyl]-2-(2-phenyl-1,3-thiazol-4-yl)-N-(pyridin-3-ylmethyl)acetamide
1-[(3-methylpyridin-2-yl)methyl]-4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
methyl 1-{[2-(methoxycarbonyl)-3-(5-methylthiophene-2-amido)thieno[2,3-b]pyridin-6-yl]methyl}piperidine-2-carboxylate
4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]benzene-1-sulfonamide
1,3-dimethyl-N-[2-(4-methylpiperazin-1-yl)propyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-4-methylphenol
N-{1-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
5-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-amine
N-(2-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
5-methyl-6-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)ethan-1-one
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-(1,3-thiazol-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-{[(2-fluorophenyl)methyl](2-methoxyethyl)carbamoyl}thiophene-2-carboxylic acid
2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-{2-[(1-cyclopentylpiperidin-3-yl)formamido]ethyl}-4-fluorobenzamide
N-(1-methoxypropan-2-yl)-1-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidine-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}piperazine
3-(4-methoxy-3,5-dimethylphenyl)-1-[3-(pyridin-4-yl)propyl]urea
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-3-(3-hydroxy-3-methylbutyl)benzamide
7-methanesulfonyl-N-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-({4-[(2,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-3-ethylpiperazin-2-one