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N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
4-ethoxy-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)propanamide
4-hydroxy-N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-4-phenylpiperidine-1-carboxamide
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxamide
N-[(3-methoxyphenyl)methyl]-3-(1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}piperidin-3-yl)propanamide
1-(4-benzylpiperazin-1-yl)-3-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}propan-1-one
2-hydroxy-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
1-(2-phenoxyethyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
3-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
9-(5-chloropyridin-2-yl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl (2S,4R)-4-cyclohexaneamido-1-[(3-ethoxy-4-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
2-{[methyl({[1-(morpholin-4-yl)cyclohexyl]methyl})amino]methyl}pyridine-3-carboxylic acid
1-[2-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-2-[2-(thiophen-2-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-1H-1,3-benzodiazole
7-(4-oxo-1,4-dihydroquinoline-2-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]propan-1-ol
4-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}-1,4-oxazepan-6-ol
1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
4-(2,6-dimethylpyridin-3-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
3-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-ethyl-N-[(4-sulfamoylphenyl)methyl]pyrimidine-5-carboxamide
(4aS,7aR)-1-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2-{4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3-thiazol-2-amine
3-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]pyridin-2-ol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
N4,N4,5-trimethyl-N2-[2-methyl-1-(pyridin-2-yl)propyl]pyrimidine-2,4-diamine
3-[(3R,4S)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2,3,4-trimethoxy-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
{2-[1-(1-benzofuran-5-carbonyl)piperidin-2-yl]ethyl}dimethylamine
(3aR,5S,6S,7aS)-2-(2-ethoxypyridine-3-carbonyl)-octahydro-1H-isoindole-5,6-diol
2,5-dimethyl-N-[3-(pyridin-3-yloxy)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-(2-fluorophenoxy)-1-(oxolane-3-carbonyl)piperidine-4-carboxylic acid
N-(2-ethoxyethyl)-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
1-{[1-(4-methylpiperazine-1-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-(4-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperazin-1-yl)ethan-1-one
2-(2-methoxyethyl)-8-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
3-{[1-(2-hydroxyethyl)piperidin-4-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-methyl-N-(4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}phenyl)methanesulfonamide
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
1-[2-(3-fluorophenyl)ethyl]-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
(2E)-3-(3,5-difluorophenyl)-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
8-[(3-methylphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-benzyl-4-(oxolane-3-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-{3-[1-(oxolan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-1,3-thiazole
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
3-(3,4-difluorophenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide