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2-(3-fluorophenoxymethyl)-N-(oxolan-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-{4-[(5-ethyl-1,3,4-oxadiazol-2-yl)amino]piperidin-1-yl}pyridine-3-carbonitrile
2-hydroxy-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
2-[4-(6-chloroquinolin-2-yl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]piperidine-3-carboxylate
3-[(3,4-dimethylphenyl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(4-methylphenoxy)ethyl]acetamide
2-[(6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrimidin-4-yl)amino]ethan-1-ol
(1S,5R)-3-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(3R,4S)-3-cyclopentaneamido-4-(propan-2-yl)pyrrolidin-1-yl]-N-methylpyridine-3-carboxamide
2-(2,5-dimethoxyphenyl)-N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
2-[1-(2-methoxyethyl)piperidin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(2-methylpropyl)-8-(2-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-4-(morpholin-4-yl)pentan-1-one
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
(3S,5R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
1-({1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}methyl)pyrrolidin-2-one
(2S,4S)-4-amino-1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzenesulfonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]pyrrolidine-2-carboxamide
N-[2-({[2-(propylsulfanyl)pyrimidin-5-yl]methyl}amino)ethyl]acetamide
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
ethyl 1-[3-({imidazo[1,2-a]pyridin-2-ylmethyl}carbamoyl)-6-(thiophen-2-yl)pyridin-2-yl]piperidine-3-carboxylate
(3R,4S)-1-[(4-methylpiperidin-1-yl)sulfonyl]-4-phenylpyrrolidin-3-amine
1-benzyl-8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aR)-5-(2,5-dimethylpyrimidin-4-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-(azepane-1-carbonyl)-1-(butan-2-yl)-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridin-4-one
1-(2-methylpropyl)-4-oxo-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
3-chloro-4-({1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-[4-(furan-2-yl)phenyl]-1-[(3-methylquinoxalin-2-yl)methyl]piperidine-3-carboxamide
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2,3-dimethylquinoxaline-6-carboxamide
5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
6-tert-butyl-1-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2,3-dimethylquinoxaline-6-carboxamide
1-(3,4-dichlorophenyl)-5-[2-(methylsulfanyl)ethyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
4-(pyridin-3-yl)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-ol
7-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
N-(2-{7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
2-{[(2-amino-6-methylpyrimidin-4-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-{[7-(piperidin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}azepan-2-one
1-cyclobutanecarbonyl-4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]piperidine
5-[(benzyloxy)methyl]-1-tert-butyl-3-(2-methoxyethyl)-1H-1,2,4-triazole
1'-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]spiro[indene-1,4'-piperidine]
4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperazine-2-carboxylic acid
1-[(3R,4R)-4-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]oxolan-3-yl]piperidine
2-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]benzoic acid
N-[(3R,4S)-4-propyl-1-[(trimethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]ethane-1-sulfonamide
N-ethyl-N-(2-hydroxyethyl)-5-methyl-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide