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(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-3-yl)methanol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[2-(methylsulfanyl)acetyl]piperidine-2-carboxamide
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N,N,4-trimethyl-3-({[3-(pyridin-3-yl)propyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(2-fluoro-3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(2-cycloheptyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
N-[(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-1H-indazole-3-carboxamide
(1S,6R)-9-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-cyclopropyl-8-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(furan-3-ylmethyl)pyrrolidin-3-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
1-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
methyl 5-(cycloheptylamino)-3-acetamido-1-ethyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methyl-2-propylpyrimidine
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-6-methylpyridine-3-carbonitrile
(3aR,6aS)-2-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-5-methyl-octahydropyrrolo[3,4-c]pyrrole
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(4-methyl-1,4-diazepan-1-yl)pyridine-3-carboxamide
(1S,4S)-2-(2,5-dimethoxyphenyl)-5-(quinoline-2-carbonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-butanamido-N,4-dimethyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
5-acetyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}thiophene-3-carboxamide
3-[4-(2,2-dimethoxyethyl)piperazine-1-carbonyl]benzonitrile
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-3-(4-chlorophenyl)propanamide
5-(4-chloro-1-methyl-1H-pyrazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-[2-(benzylamino)ethyl]-1-[2-(3,4-dimethoxyphenyl)ethyl]pyrrolidin-2-one
N-(4H-1,2,4-triazol-4-yl)-2,1-benzoxazole-3-carboxamide
N-{4-[4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)piperidin-1-yl]phenyl}cyclopentanecarboxamide
2-methoxy-3-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}pyridine
2-methyl-7-(2,3,4-trimethoxybenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-{4-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazin-1-yl}pyrazine
1-(2-methoxyethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
4-hydroxy-2-methyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}pyrimidine-5-carboxamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}hexan-1-one
N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
2-(2-chloro-4-fluorophenoxymethyl)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
N-(2-oxopiperidin-3-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(4-methyl-5-phenylthiophen-2-yl)formamido]acetic acid
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2,4-dimethylpyrimidine-5-carboxamide
methyl 4-{3-[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)amino]propanamido}benzoate
N4-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-6-(morpholin-4-yl)pyrimidine-2,4-diamine
2-{4-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}phenol
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-phenoxyacetamide
(4S)-3-(2-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-oxoethyl)-4-phenyl-1,3-oxazolidin-2-one
5-acetyl-N-(1-benzothiophen-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[(2-phenoxypyridin-3-yl)methyl]-2-(1H-pyrazol-1-yl)propanamide
2-(dimethylamino)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(4-methylphenyl)acetamide
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide