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2-ethyl-N-[(5-methylpyrazin-2-yl)methyl]pyrimidine-5-carboxamide
2-({[4-(methylsulfanyl)phenyl]methyl}({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})amino)ethan-1-ol
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(isoquinolin-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-methyl-4-phenyl-1,3-thiazole-5-carboxamide
2-{9-[2-(4-methoxyphenyl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(2-ethoxyphenyl)methyl]pyrrolidin-3-yl]methanol
1-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-(pyridin-3-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
ethyl 4-(2-{[4-(1H-pyrazol-1-yl)phenyl]carbamoyl}piperidin-1-yl)piperidine-1-carboxylate
2-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(3,4-difluorophenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
3-[(dimethylamino)methyl]-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]pyrrolidin-3-ol
3-(2H-1,3-benzodioxol-5-yl)-1-ethyl-N,N-dimethyl-1H-1,2,4-triazol-5-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
(1R,3S)-1-hydroxy-3-methoxy-N-(4-methylphenyl)-7-azaspiro[3.5]nonane-7-carboxamide
3-({1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}oxy)pyridine
3-{2-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]ethyl}-5-ethyl-1,2,4-oxadiazole
3-{5-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-[4-(propan-2-yl)morpholin-2-yl]-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]morpholine-4-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(2-methylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 4-(5-{[2-(2-hydroxyethyl)-3-oxopiperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-(2-fluorophenyl)-N-[2-(morpholine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-{1-[5-(4-chlorophenyl)-1,2,4-triazin-3-yl]piperidin-4-yl}-5-methyl-1H-1,3-benzodiazole
(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)(2-methoxyethyl)(pyridin-3-ylmethyl)amine
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-2-one
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-cyclopentyl-6-oxo-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-ethyl-4-{[4-(quinazolin-4-yl)piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
3-[(2,5-difluorophenyl)methyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[4-(oxan-2-ylmethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl]methanol
4-({[1-methyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)benzene-1-sulfonamide
1-(azepan-1-yl)-3-[3-(morpholin-4-ylmethyl)phenoxy]propan-2-ol
3-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-1,2-dimethyl-1H-indol-5-ol
2-[2-(1H-imidazol-4-yl)ethyl]-8-(2-methoxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopentyl-N-methyl-N-[3-(3-methylphenoxy)propyl]-5-oxopyrrolidine-3-carboxamide
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(3-phenylpropyl)benzamide
1-({4-[4-methoxy-4-(prop-2-en-1-yl)piperidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)-1H-1,3-benzodiazole
(2R,6R)-4-(1H-imidazol-2-ylmethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{[5-(1-cyclobutanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
N,N-diethyl-4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}aniline
4-(4-chlorophenyl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)butanamide
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
2-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-ethylacetamide
8-[(3-ethoxy-4-hydroxyphenyl)methyl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione