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4-[(benzyloxy)methyl]-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(4-fluorophenyl)methyl]-1-[2-({[4-(propan-2-yl)phenyl]methyl}amino)ethyl]-1H-1,2,3-triazole-4-carboxamide
(5-{1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)methanol
7-methyl-2-[2-(naphthalen-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-[(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)methyl]benzene-1,2-diol
(2S,4S)-4-amino-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]pyrrolidine-2-carboxylic acid
4-[5-(5-chloro-6-oxo-1,6-dihydropyridin-3-yl)-3-methyl-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
methyl 3-{[(2-fluorophenyl)formamido]methyl}-5-(2-methoxybenzamido)benzoate
4-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
4,6-dimethyl-N-(1-methylpiperidin-4-yl)-2-oxo-N-(pyridin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
1'-[3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]spiro[indene-1,4'-piperidine]
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]propanamide
N,N-dimethyl-6-{3-[1-(pyridin-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrazine-2-carboxamide
1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(furan-2-yl)-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]azepane-1-carboxamide
2-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-6-methylquinolin-4-ol
2-{[4-(3-methoxyphenyl)-5-(1H-pyrazol-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-(3-fluoropyridin-4-yl)-2-(6-methoxynaphthalen-2-yl)morpholine
(4aR,7aS)-1-(2-hydroxyethyl)-4-[3-(4-hydroxyphenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-(2-chlorophenyl)cyclopropyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-methyl-1-(naphthalen-1-ylmethyl)-N-(pyrazin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
N-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrimidin-2-amine
(5S,9aS,9bS)-5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
1-methyl-4-{4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}piperazine
3-(4-{[2-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)propanamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-1-yl]acetamide
N-(1-cycloheptylpiperidin-3-yl)-2-(2-oxopiperidin-1-yl)acetamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
1-cyclopropyl-3-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(thiomorpholin-4-yl)pyridine-3-carboxamide
(2R,6S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
(1S,6R)-9-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(thiophen-2-yl)propan-1-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-(4-{4-[ethyl(methyl)amino]pyrimidin-2-yl}piperazin-1-yl)-6-methylpyrimidin-2-amine
methyl (2S)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]piperidine
4-{1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-tert-butyl-N-[(3,5-difluoro-4-methoxyphenyl)methyl]-4-hydroxypyrimidine-5-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(1,4-dioxan-2-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-ethoxypropan-1-one