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N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
5-methyl-1-{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-(1-methylpiperidin-2-yl)-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}propanamide
6-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1,2-dihydropyridin-2-one
1-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1H-indole-3-carboxamide
3-methyl-8-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[4-(6-methyl-2-phenylpyrimidin-4-yl)piperazin-1-yl]pyrazine-2-carbonitrile
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-6-cyclopropylpyrimidin-4-amine
3-methoxy-N-[1-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
1-(2-{[1-(4-methoxyphenyl)piperidin-4-yl]amino}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
2-[(4-chlorophenyl)methyl]-8-[(4-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
8-fluoro-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]quinoline-2-carboxamide
5-acetyl-2,4-dimethyl-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]-1H-pyrrole-3-carboxamide
(1R,9S)-5-amino-3-(furan-3-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
3-[(3R,4S)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2,4-dimethyl-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide
2-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-4-(pyridin-4-yl)pyrimidin-2-amine
(3S,4R)-1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}[2-(1H-imidazol-4-yl)ethyl]amine
1-[6-(3-methylphenyl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}propanamide
2-(azepan-1-yl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)acetamide
4-phenyl-N-(1-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-hydroxy-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)(pyridin-2-yl)methanol
(2R,3R)-3-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-methylurea
methyl 4-[5-({7-ethyl-2,7-diazaspiro[4.4]nonan-2-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
5-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]thiophene-2-carboxylic acid
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
5-[4-(4-chlorophenyl)piperazine-1-carbonyl]-1-cyclopentylpiperidin-2-one
1-(oxolan-3-ylmethyl)-4-phenoxypiperidine-4-carboxylic acid
[3-(1H-indazol-1-yl)propyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
1-ethyl-4-{[3-(2-propylpyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperazine
4,6-dimethyl-N-{3-[methyl(phenyl)amino]propyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(1S,5R)-6-propyl-3-[(2,4,6-trimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-cyclopropanecarbonyl-1'-(3,4-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
6,7-dimethoxy-2-[4-(pyridin-4-yl)pyrimidin-2-yl]-1,2,3,4-tetrahydroisoquinoline
3-(1-methyl-1H-pyrrol-2-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
2-cyclopentyl-N-(3-methoxypropyl)-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
3-[(3R,4S)-4-(dimethylamino)-1-[3-(3-methoxy-4-methylphenyl)propanoyl]piperidin-3-yl]propanoic acid
(1S,5R)-1,3,3-trimethyl-N-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-6-azabicyclo[3.2.1]octane-6-carboxamide
N-cyclohexyl-N-(2-hydroxyethyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
[(2,4-difluorophenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
5-(3-methylfuran-2-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid