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2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-(4-methoxyphenyl)-5-methylpyridine-3-carbonitrile
(4aS,8aS)-2-cyclohexanecarbonyl-7-(pyridin-4-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
3-[1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]-N-phenylpropanamide
(3aR,6aR)-2-cyclohexyl-5-(5-methyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}morpholine
2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methylacetamide
N-[2-(2-chloro-6-fluorophenyl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
methyl (2S)-3-methyl-2-({5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazol-3-yl}formamido)butanoate
3-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
1-(carbamoylmethyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidine-4-carboxamide
1-[3-(1H-imidazol-1-yl)propyl]-5-(2-methoxy-4-methylphenyl)-4-phenyl-1H-imidazole
6-(benzyloxy)-4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
1-(3-chloro-5-fluorophenyl)-3-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}urea
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
N-[(2S)-2-aminopropyl]-2-(4-tert-butylphenoxymethyl)-4-hydroxypyrimidine-5-carboxamide
2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]propane-1,3-diol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-cycloheptyl-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-cyclopropyl-1H-1,2,4-triazole
2-{4-[(2,2-difluoro-2H-1,3-benzodioxol-4-yl)methyl]morpholin-3-yl}acetic acid
2-cyclohexyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(3-methylbutyl)-8-[3-(thiophen-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3,3-dimethyl-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(morpholin-4-ylmethyl)piperidin-4-ol
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)methylamine
methyl 3-(2-chloro-6-fluorobenzamido)-6-[(3-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
2,6-dimethyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-4-carboxamide
N-methyl-N-(oxan-4-ylmethyl)-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[2-(4-fluorophenyl)azetidin-1-yl]ethan-1-one
4-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]-1,4-oxazepan-6-ol
2-methoxy-N-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(naphthalen-1-ylmethyl)pyrrolidin-3-yl]methanol
1-cyclopropyl-3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[(3-methylthiophen-2-yl)methyl]urea
7-[(4-phenylpiperazin-1-yl)methyl]-4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-4-(3-chloro-4-hydroxy-5-methoxyphenyl)-6-cyclobutylpyridine-3-carbonitrile
(3R,4R)-4-cyclobutyl-1-(5,6-dimethylpyrazin-2-yl)-3-methylpiperidin-4-ol
methyl 2-(azepane-1-sulfonyl)-6-[3-(methylsulfanyl)propyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-cyclohexyl-N-{[3-(trifluoromethoxy)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
1-[3-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-[3-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(3-methyloxetan-3-yl)methyl]benzamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]pyridine-3-sulfonamide
1-[6-(cyclopropylmethoxy)-4-[(3-methoxyphenyl)methyl]-3-oxo-1,4-diazepan-1-yl]-3-phenylpropane-1,2-dione
1-(2-methylfuran-3-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-{1-[1-(3-chloro-4-fluorobenzoyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-(5-propyl-1,2-oxazole-4-carbonyl)-7-azaspiro[3.5]nonan-1-ol
5-(1-{[4-(dimethylamino)phenyl]methyl}piperidin-4-yl)-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione