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7-[(2,3-difluorophenyl)methyl]-2-(propane-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
[(3-fluorophenyl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
5-{2-[2-(cyclooctylamino)ethyl]morpholin-4-yl}-2-methyl-2,3-dihydropyridazin-3-one
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}butan-1-one
3-[5-(2,3-difluoro-6-methoxybenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-chloro-1-ethyl-N-(3-phenylprop-2-yn-1-yl)-N-propyl-1H-pyrazole-5-carboxamide
4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-1-(3-phenylbutyl)piperidine
1-{1-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(oxan-4-ylmethyl)benzamide
5-benzenesulfonamido-1-ethyl-2-methyl-N-[2-(methylsulfanyl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
(2E)-3-(3,5-difluorophenyl)-1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
3-methoxy-1-{1-methyl-4-propyl-1,4,9-triazaspiro[5.5]undecan-9-yl}propan-1-one
butyl 3-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]carbamoyl}piperidine-1-carboxylate
ethyl 4-({cyclopentyl[(3-methylthiophen-2-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylate
6-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,4-oxazepan-6-ol
N-cyclohexyl-N-(2-hydroxyethyl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-(4-fluorophenyl)-4-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]piperazine
4-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1-[2-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole
{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[1-(thiophen-2-yl)propan-2-yl]amine
(7R,8aS)-7-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-2-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-benzyl-N-(2-oxoazepan-3-yl)-1,3-thiazole-4-carboxamide
4-(4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}phenyl)-2-methylbutan-2-ol
1-(furan-3-carbonyl)-3-(3-methylphenyl)piperidine
1-ethyl-5-methyl-N,N-bis(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-3-yl]methanol
[1-(1-{5-cyclopropyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)piperidin-3-yl]methanol
3-{2-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
[(3-{2-[1-(2,4-dimethoxybenzoyl)piperidin-2-yl]ethoxy}phenyl)methyl](methyl)(quinolin-8-ylmethyl)amine
3-ethyl-6-[4-(2,2,2-trifluoroethyl)piperazine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
5-({[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-1,3,4-thiadiazol-2-amine
1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(6-methylpyridin-2-yl)piperazine
3-[4-(2-methoxyphenyl)piperazin-1-yl]-N-(4-methylphenyl)piperidine-1-carboxamide
4-(4-chlorophenyl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]butan-1-one
N-[(3S,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(4aS,8aS)-2-cyclopentanecarbonyl-7-(pyridine-4-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
3-(1,4-diazepane-1-carbonyl)-N-(thiophen-3-ylmethyl)benzene-1-sulfonamide
N-[3-(methylsulfanyl)propyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-chloro-4-hydroxy-N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
1-[2-(dimethylamino)-6-(2-methylphenyl)pyridine-3-carbonyl]piperidin-4-ol
2-(2-phenylethyl)-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-4-{[methyl({[5-(pent-2-yn-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl})amino]methyl}pyrrolidin-2-one
N-ethyl-5-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]pyrimidin-2-amine
6-methoxy-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-cyclopropyl-3-[(4-fluorophenyl)methyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-[(5-methylthiophen-2-yl)methyl]piperidine
2-(5-methyl-1H-pyrazole-3-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
2-ethoxy-4-[({[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenol
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide