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2-[(3,4-dimethoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]-1,3-benzoxazole-6-carboxamide
1-({2-[3-(azepan-1-yl)-2-hydroxypropoxy]-5-chlorophenyl}methyl)piperidin-4-ol
4-(2-methoxyphenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,2-dimethylcyclopropane-1-carboxamide
3-benzyl-4-(3-fluoro-4-methylbenzoyl)piperazin-2-one
methyl 1-({[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}carbamoyl)cyclopropane-1-carboxylate
1-[(2E)-but-2-en-1-yl]-4-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-1,4-diazepane-6-carboxylic acid
N-(1-ethyl-1H-pyrazol-4-yl)-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
N4-[1-(thiophen-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-3-(1H-1,2,3,4-tetrazol-5-yl)urea
N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)quinoxaline-5-carboxamide
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-(4-methyl-3-phenyl-1H-pyrazol-1-yl)acetamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-benzyl{[3-(1H-pyrazol-5-yl)phenyl]amino}sulfonamide
5-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
6-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
(2R,3R,6R)-5-(2-ethylpyrimidine-5-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2-methylphenyl)-3-{2-oxo-2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
N-(4-chloro-2-methylphenyl)-3-[4-(methylsulfanyl)benzoyl]piperidine-1-carboxamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)cyclohexanecarboxamide
6-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-cyclopentyl-6-oxo-N-[2-(2-oxopiperidin-1-yl)ethyl]piperidine-3-carboxamide
3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-N-[2-(pyridin-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-2-one
4-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-2-(propan-2-yl)-1,3-oxazole
2-[1-(4-chlorophenyl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[2-(5-methylfuran-2-yl)ethyl]acetamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(3-methoxyphenyl)methyl]piperazine
1-benzyl-N-cyclopropyl-N-(1,3-thiazol-5-ylmethyl)-1H-pyrazole-4-carboxamide
2-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]-3-methylquinoxaline
methyl 2-[(2-methoxyethyl)sulfamoyl]-6-[(3-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
3-[3-(propan-2-yloxy)benzoyl]-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]benzonitrile
[3-(cyclopropylmethyl)-1-(5-ethylthiophene-2-carbonyl)piperidin-3-yl]methanol
8-[3-(2-methyl-1H-indol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(4-methylbenzenesulfonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-fluoroethyl)-3-{[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]sulfamoyl}benzamide
5-[({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
4-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}pyridine
4-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-{3-[(benzylsulfamoyl)amino]propyl}-N-methylaniline
4-(1H-pyrazol-3-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]benzamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(3-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(3-methylpyridin-4-yl)methyl]acetamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
methyl 4-[({2-[5-oxo-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-2-yl]ethyl}amino)methyl]benzoate