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2-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}benzoic acid
1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
1-(3-chlorophenyl)-4-(4-fluoro-3-methylbenzoyl)piperazin-2-one
2-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
1-{4-[(tert-butylamino)methyl]-2-methoxyphenoxy}-3-(morpholin-4-yl)propan-2-ol
8-[3-(methylsulfanyl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
N5,N5-dimethyl-N6-(quinolin-6-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]-3-(pyridin-3-yl)propan-1-one
(2S,6S)-1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-({1-[ethyl(methyl)amino]cyclopentyl}methyl)-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-(3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
5-[(2,5-dimethoxyphenyl)methyl]-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3R,5S)-N3-(4-fluorophenyl)-N5-[(4-fluorophenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
4-ethyl-1-methyl-3-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-ethyl-3-{1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
N-methyl-N-[2-phenyl-1-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]oxane-4-carboxamide
11-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecane
N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
3-methoxy-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
N-[(5-methylfuran-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[(cyclopropylmethyl)sulfanyl]-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
1-(methoxymethyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]cyclobutane-1-carboxamide
3-(4-{[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}phenyl)prop-2-yn-1-ol
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-4-yl)ethyl]amine
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-[(4-methoxy-3-methylphenyl)methyl]-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-butyl-1-methyl-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazin-2-one
(3S,4S)-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
[5-(1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)furan-2-yl]methanol
4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-phenylpiperazine-2-carboxylic acid
4-(2-{1-[(2,6-difluoro-3-methylphenyl)methyl]piperidin-2-yl}ethyl)morpholine
(1S,5R)-3-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(1H-imidazol-1-ylmethyl)-1-[(3-phenoxyphenyl)methyl]piperidin-4-ol
N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
2-(2-methoxyethyl)-6-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,3-benzoxazole
5-({[(3-{2-[4-(3,5-dimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
2-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,3-benzoxazole-6-carboxamide
1-(4-fluorophenyl)-4-[6-methoxy-3-oxo-4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]butane-1,4-dione
3-(1-methyl-1H-indazol-5-yl)-1-{[1-(morpholin-4-yl)cyclohexyl]methyl}urea
N-(cyclopropylmethyl)-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2,3-dimethyl-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-1H-indole-5-carboxamide
[(2-fluorophenyl)methyl](2-methoxyethyl){[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}amine
2,3,5-trimethyl-N-[3-(methylsulfanyl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
(4aR,8aR)-2-cyclobutanecarbonyl-7-[2-(2-ethylphenoxy)ethyl]-decahydro-2,7-naphthyridin-4a-ol
N-methyl-3-(4-methyl-1H-pyrazol-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide