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N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(3-methoxyphenyl)acetamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[5-(2,3-dihydro-1H-inden-2-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
N-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-benzenesulfonamido-1-ethyl-N-[(3-methoxyphenyl)methyl]-2-methyl-1H-1,3-benzodiazole-7-carboxamide
N3-cycloheptyl-N5-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(3-methoxyphenyl)-1-[1-(2-phenylpropanoyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
3-{5-[(3,4-dimethoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-(piperidin-4-yl)urea
1-(4-phenylpiperazin-1-yl)-3-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]propan-1-one
N-methyl-2-oxo-1-phenyl-N-(quinolin-2-ylmethyl)pyrrolidine-3-carboxamide
N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
1-[1-(furan-2-ylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanamide
1-(2-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
N,N-dimethyl-3-{[(2S,5R)-5-(thiomorpholin-4-ylmethyl)oxolan-2-yl]methyl}benzamide
N3-(2-methoxyethyl)-N5-[(1R)-1-(3-methoxyphenyl)ethyl]-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
benzyl({[4-(1H-pyrazol-4-yl)phenyl]methyl})amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(dimethyl-1,3-thiazol-5-yl)-N-methylacetamide
3-(1-{2-[(cyclopropylmethyl)sulfanyl]acetyl}piperidin-3-yl)benzoic acid
1-(3-phenylpropyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepane
N-ethyl-1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidine-3-carboxamide
2-[3-(dimethylamino)pyrrolidin-1-yl]-1-[3-(2-ethylphenoxy)azetidin-1-yl]ethan-1-one
2-(dimethylamino)-N-ethyl-2-(3-fluorophenyl)-N-(2-methoxyethyl)acetamide
N-ethyl-2-methyl-N-(oxan-4-ylmethyl)-6-(piperidin-4-yl)pyrimidin-4-amine
3-[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
9-(2-hydroxy-3-methylbenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-4-(trifluoromethoxy)benzene-1-sulfonamide
1-ethyl-3-(4-methylpiperazine-1-carbonyl)-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-(2-chloro-6-methoxyphenyl)pyridine-3-carbonitrile
1-(3-methoxyphenyl)-4-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
6-{4-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperazin-1-yl}-9H-purine
2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[4-(thian-4-yl)piperazin-1-yl]ethan-1-one
1-(furan-2-carbonyl)-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-N-[3-(propan-2-yloxy)propyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})(pyridin-3-ylmethyl)amine
3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}propanamide
6-methoxy-1-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1H-indole-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-4-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidin-3-yl}pyridine
N-butyl-N-methyl-3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-(4-methylpiperidine-4-carbonyl)piperidine
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
4-cyclobutyl-6-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrimidin-2-amine
1-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
5-benzyl-1-(cyclopropylmethyl)-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[(4-chlorophenyl)methyl]-5-{3-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
methyl 3-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate