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N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)cyclopropanecarboxamide
2-[(adamantan-1-ylmethyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino]ethan-1-ol
1-cyclopentyl-3-[2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-oxoethyl]-3-(3-fluorophenyl)pyrrolidine-2,5-dione
(5S,9aS,9bS)-5-(1,5-dimethyl-1H-pyrazol-4-yl)-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{[5-(2-fluorophenyl)furan-2-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
3-(4-acetylphenyl)-1-[3-(cyclohexyloxy)propyl]urea
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(3-methylbutyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-{[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]methyl}cyclopropanamine
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-3-(pyridin-3-yl)propanamide
methyl 3-(2-cyclohexylacetyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl[1-(pyrimidin-4-yl)ethyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
6-(4-chlorophenyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
dimethyl({[(3S,4R)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
(1S,5R)-N-cyclopentyl-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(butan-2-yl)[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](pyridin-4-ylmethyl)amine
9-(cyclopropylmethyl)-1-methyl-4-(5-propyl-1,3,4-thiadiazol-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}propanamide
5,5-dimethyl-3-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-1,3-oxazolidine-2,4-dione
N-[(3-methylthiophen-2-yl)methyl]-3-propyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
methyl[(3-phenyl-1H-pyrazol-5-yl)methyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
4-{2-[1-(cyclopropylmethyl)piperidin-2-yl]ethyl}phenol
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}propanamide
9-ethyl-1-methyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-methyl-4-phenyl-9-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-2,9-diazaspiro[5.5]undecane
2-(2,3-dihydro-1H-isoindol-2-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]oxane-4-carboxamide
N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-1-benzothiophene-5-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(pyridin-4-yl)ethyl]piperidin-2-one
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-4-(piperidin-3-yl)benzamide
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-methylpyrimidin-4-amine
(3R,4R)-1-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
2-{5-methyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl}benzoic acid
1-(4-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenyl)ethan-1-one
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[3-(morpholin-4-yl)propyl]amine
2-(cyclopropylmethyl)-N-[1-(3-methylpyridin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4R)-1-[3-(dimethylamino)benzoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-{2-[3-(ethoxymethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
ethyl 1-(oxolane-3-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylate
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-4-(pyridin-4-yl)pyrimidin-2-amine
2-amino-8-(5-chloro-2,3-dimethoxyphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-(6-methylpyridine-2-carbonyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-3-(6-oxo-1,6-dihydropyridazin-3-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
(2E)-3-(4-methoxyphenyl)-1-{4-[3-(thiomorpholin-4-ylmethyl)phenoxy]piperidin-1-yl}prop-2-en-1-one
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-oxo-1,2-dihydroquinoline-3-carboxamide
1-{3-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]phenyl}-5-methyl-1H-1,2,3,4-tetrazole
methyl 3-[2-(4-acetylphenoxy)acetyl]-9-(cyclopentyloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate