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3-{2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
6-methoxy-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrimidin-4-amine
1-(2-methylbutyl)-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(thian-4-yl)piperazin-2-yl}ethan-1-ol
3-{2-[2-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
N-({5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
3-{[5-(3-fluorophenyl)-1,2,4-triazin-3-yl](methyl)amino}-1-phenylpropan-1-ol
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}benzonitrile
1-(4-fluorophenyl)-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butan-1-one
2-(1-ethyl-1H-pyrazol-4-yl)-3,6-dimethyl-4-(4-methylpiperidine-1-carbonyl)quinoline
4-(2-methoxy-5-methylphenyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazole
1-cyclopentanecarbonyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpiperidine-4-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(3-methylphenyl)acetamide
methyl 3-(furan-2-amido)-5-{[(3-methoxyphenyl)formamido]methyl}benzoate
5-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2-methyl-1-benzofuran-7-amine
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
2-[3-(methylsulfanyl)propanoyl]-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-methyl-5-{[(3-methyloxetan-3-yl)methyl]amino}-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[(3-methoxypiperidin-1-yl)methyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methylpiperidin-4-ol
2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-6-({1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}methyl)-1,2-dihydropyridine-3-carboxamide
2-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-benzoyl-4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
(1R,5R)-6-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-5-[2-oxo-2-(pyridin-3-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
6-methoxy-4-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
4-(4-ethoxy-3-methylphenyl)-N-methyl-4-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)butanamide
(3S,4S)-4-cyclopropyl-1-{2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}pyrrolidine-3-carboxylic acid
2-{[(3S,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-(cyclohexylmethyl)pyrrolidin-3-yl]sulfanyl}-4,6-dimethylpyrimidine
4-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
methyl 3-[2-(4-chlorophenoxy)acetyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-2-one
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
6-(3-fluoro-4-methoxyphenyl)-N-[(5-methylthiophen-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-(ethylamino)-N-[(2-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(2-amino-5-ethylpyrimidin-4-yl)amino]-3-(dimethylamino)propan-2-ol
1-[3-fluoro-5-(trifluoromethyl)phenyl]-3-[1-(methoxymethyl)cyclopropyl]-3-methylurea
2-(2-{1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(2S,4S)-4-amino-N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-1-methylpyrrolidine-2-carboxamide
N,N,8-trimethyl-2-[1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-ethyl-N,4-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-oxazole-5-carboxamide
6-fluoro-4-[1-(3-methylpyridin-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinolin-2-one
ethyl 2-(2-{[5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazol-4-yl]formamido}ethyl)-1,3-thiazole-4-carboxylate
1-{5-[(4-methylpiperazin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}azocane
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(3-phenylphenyl)methyl]acetamide
(1-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-yl)methanol
3-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-9-methoxy-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide