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1-phenyl-N-({1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-3-yl}methyl)methanesulfonamide
2-{[7-(2-methyl-5-propylpyrimidin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}propan-1-ol
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
5-methanesulfonamido-1-(2-phenylethyl)-N-[3-(pyridin-3-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-methylbutan-1-one
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[3-(methylsulfanyl)propyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-{3-oxo-3-[2-(2-phenylethyl)piperidin-1-yl]propyl}piperidin-2-one
N-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-N-[(3-methylthiophen-2-yl)methyl]cyclopropanamine
2-[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]-6-methylpyridine-3-carbonitrile
6,7-dimethoxy-2-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
4-(4-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
N-cyclopropyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)pyridine-2-carboxamide
2-cyclopentyl-N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)acetamide
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
(2S)-2-(methoxymethyl)-N-(4-methoxynaphthalen-2-yl)pyrrolidine-1-carboxamide
2-(5-fluoro-2-methoxyphenyl)-2-[(furan-2-ylmethyl)(pyridin-4-ylmethyl)amino]acetic acid
1-(furan-3-carbonyl)-4-(1H-indol-2-ylmethyl)-1,4-diazepan-6-ol
4-cyclobutanecarbonyl-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
4-[(4-fluorophenyl)methyl]-1-[2-(2-hydroxyethoxy)ethyl]-3-(propan-2-yl)-1,4-diazepan-5-one
[(1-methyl-1H-pyrazol-4-yl)methyl]({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})(propan-2-yl)amine
N-cyclopropyl-6-(2-methoxyphenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)propanamide
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-{5-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-4-methylpiperazine
N-[(3-chlorophenyl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(1,3-thiazol-4-yl)phenyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
2-(1-cyclohexyl-4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
6-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-5,6-dihydro-1,6-naphthyridin-5-one
methyl 4-methoxy-3-{[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]amino}benzoate
methyl[2-(oxan-4-yl)ethyl]{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
2-{[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
(1-{3-[4-(1H-imidazol-1-ylmethyl)phenyl]phenyl}ethyl)dimethylamine
8-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({5-[(5-chlorothiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-[3-(3-methylphenyl)propyl]-4-(piperidin-3-yl)benzamide
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
ethyl 1-(1-{4-[(2H-1,3-benzodioxol-5-ylmethyl)carbamoyl]phenyl}piperidin-4-yl)piperidine-4-carboxylate
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]butanamide
1-[(2-methylphenyl)methyl]-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
3-(but-2-yn-1-yl)-5-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
1-benzoyl-N-(isoquinolin-5-ylmethyl)-N-methylpiperidin-4-amine
1'-[2-(methylamino)pyridine-4-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(3-methoxyphenyl)-3-[1-(quinolin-8-ylmethyl)piperidin-4-yl]propanamide
2-methyl-N-[2-(7-methyl-1H-indol-3-yl)ethyl]-6-(piperidin-4-yl)pyrimidin-4-amine
N-ethyl-5-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)pyrimidin-2-amine
3-(4-cyanopiperidine-1-carbonyl)-N-(oxolan-3-ylmethyl)benzene-1-sulfonamide