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{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-butyl-N-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
methyl 2-{N-methyl-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}acetate
N-[(3S,4R)-1-[(2-fluorophenyl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-[(5-methylpyrazin-2-yl)methyl]benzamide
2-{[4-(2,5-dimethylphenyl)piperazin-1-yl]methyl}-4-(pyridin-2-yl)phenol
2-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-4,5,6-trimethylpyridine-3-carbonitrile
N-(2-{7-[(2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-3-fluoropyridine-4-carboxamide
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}oxolane-3-carboxamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
4-phenyl-N-(1-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
4-hydroxy-1-(5-propyl-1,2,4-oxadiazol-3-yl)piperidine-4-carboxylic acid
N-(1-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(2-methylphenyl)piperazin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
5-{1-[(3E)-hex-3-enoyl]pyrrolidin-2-yl}-N-(3-hydroxyphenyl)thiophene-2-carboxamide
2,4-dimethyl-N-[4-(4-{[2-(propan-2-yloxy)ethyl]amino}piperidin-1-yl)phenyl]benzamide
N-(4-aminobutyl)-3-(4-methylphenyl)-3-phenylpropanamide
8-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
(4aS,8aR)-1-butyl-6-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-[4-(hydroxymethyl)phenyl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
1-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
(4aR,7aS)-1-(2-{methyl[2-(pyrrolidin-1-yl)ethyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(2-fluoro-4-methoxyphenyl)-2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
4-[4-(2-ethyl-1H-imidazol-1-yl)phenyl]-1,3-thiazol-2-amine
8-(4-methylquinolin-2-yl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(4aS,8aR)-1-(2-phenylethyl)-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridin-2-one
2-[3-fluoro-5-(trifluoromethyl)phenyl]pyridine-4-carboxamide
5-{cyclopropyl[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1-methyl-1H-1,2,4-triazole
N-[(2-ethoxypyridin-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}azepane
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
(1R,5R)-3-methanesulfonyl-6-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)methanol
2-[9-(furan-3-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
3-chloro-N-[4-(4-{[(1-ethylpyrrolidin-2-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
1-(furan-2-ylmethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]piperidine-4-carboxamide
(4aS,8aS)-2-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-decahydroisoquinolin-4a-ol
3-({5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)benzonitrile
N-(cyclohexylmethyl)-4-({4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carboxamide
1-(4-fluorophenyl)-4-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]butane-1,4-dione
4-benzyl-3-ethyl-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1,4-diazepan-5-one
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(dimethyl-1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[2-(2-oxopyrrolidin-1-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one