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(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1H-imidazol-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
5-{2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-chloro-4-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]benzamide
5-[(isoquinolin-5-yloxy)methyl]-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
2-ethyl-9-(2-methylbenzenesulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-hydroxy-2-phenylethan-1-one
N-(5-oxo-1-phenylpyrrolidin-3-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N2,N2,5,6-tetramethyl-N4-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidine-2,4-diamine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-9-oxo-9,10-dihydroacridine-4-carboxamide
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(3-ethoxy-4-hydroxyphenyl)pyridine-3-carbonitrile
1-cyclopentyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-6-oxopiperidine-3-carboxamide
3-(4-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1H-pyrazol-5-ol
N-({1-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
4-[4-({imidazo[1,2-a]pyridin-3-ylmethyl}amino)piperidin-1-yl]-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-[3-(propan-2-yloxy)benzoyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
1-{4-[3-(4-methoxy-2-methylbenzoyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-(4-methylpiperazin-1-yl)propan-1-one
(4aS,8aR)-6-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-(3,4-dimethylphenyl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
[2-({4-[(2,3-difluoro-4-methylphenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
6-(2-chlorophenyl)-N-(2-hydroxybutyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
3-(1H-1,2,3-benzotriazol-5-yl)-1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}urea
4-[({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amino]-1-phenylpyrrolidin-2-one
5-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-N-propylpyrimidin-2-amine
4-ethyl-1-methyl-3-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(1H-imidazol-1-ylmethyl)-1-[4-(5-methylfuran-2-yl)benzoyl]piperidine
N-[2-(quinolin-6-ylmethyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
2,6-dimethyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-{[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1,3-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}quinoline-4-carboxylic acid
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-3-[4-(4-methylphenyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
8-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
N-[2-methyl-5-({[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}amino)phenyl]propanamide
(1S,5R)-6-benzyl-3-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
4-[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl]-1-cyclopentylpiperazin-2-one
5-[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrazin-2-ol
N-[phenyl(pyridin-4-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(propan-2-yloxy)ethyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(4aR,7aS)-4-[(4-methoxy-3-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[5-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol