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{[(1R,5S,6S)-3-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
3-[3-(methoxymethyl)piperidin-1-yl]-5-(naphthalen-1-yl)-1,2,4-triazine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-{4-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]piperidin-1-yl}pyrimidine
2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
4-[2-(1H-pyrazol-1-yl)ethyl]-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
N,2-dimethyl-N-(2-phenoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-cyclobutyl-3-(2-fluorophenyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
12-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-15-methyl-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
N-[3-(2,5-dimethylphenoxy)propyl]-4-hydroxy-N,2-dimethylpyrimidine-5-carboxamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)cyclopropanecarboxamide
7-methyl-4-(piperidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
3,3,3-trifluoro-N-[(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
methyl 4-(5-{[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-cyclohexyl-3-hydroxy-4-(3-methyl-1,2-benzoxazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{4-cyclobutyl-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(3R,4S)-4-cyclopropyl-1-(1,2-dimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-amine
4-{1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperidin-4-yl}pyridine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]acetamide
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethyl-4-oxobutanamide
3-[2-(4-chlorophenyl)acetyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-cyclopropyl-4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]pyrrolidin-2-one
3-(3,4-difluorophenyl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
(2S,4R)-4-(cycloheptylamino)-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-(2-oxopyrrolidin-3-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2R)-2-amino-3-hydroxy-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
2-{1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]pyrrolidin-3-yl}benzoic acid
1-{5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-{[({2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}methyl)amino]methyl}-1,2-dihydrophthalazin-1-one
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]pyrrolidin-3-yl]methanol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)benzamide
N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1H-imidazole-2-carboxamide
5-(7-{[4-(benzyloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)pyrrolidin-2-one
methyl 2-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}benzoate
2-{4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-1-yl}pyridine-3-carboxamide
5-(1H-imidazol-2-yl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]thiophene-2-carboxamide
2,4-dimethyl-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)pyrimidine
1-(2-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
3-(4-methoxyphenyl)-N-methyl-N-[2-(2-oxopiperidin-1-yl)ethyl]-3-phenylpropanamide
4-(2-methoxyacetyl)-N-[3-(prop-2-en-1-yloxy)phenyl]-1,4-diazepane-1-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-(2-methoxy-6-methylbenzoyl)piperazin-2-one
2-ethyl-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide
{5-[2-(4-chlorophenyl)morpholine-4-carbonyl]furan-2-yl}methanol
N,N-dimethyl-2-[(3-{[2-(1H-pyrazol-4-yl)ethyl]sulfamoyl}phenyl)formamido]acetamide
methyl 4-[2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-3-cyanopyridin-4-yl]-1H-pyrazole-3-carboxylate
N-[2-(2-phenoxyethoxy)phenyl]-3-(propan-2-yl)-1H-pyrazole-4-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(4-methyl-1,3-oxazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one