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[(2-{[5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenyl)methyl]dimethylamine
methyl 1-{[6-methyl-4-(thiomorpholin-4-yl)quinazolin-2-yl]methyl}piperidine-2-carboxylate
N-methyl-2-[3-oxo-1-(2-oxobutanoyl)piperazin-2-yl]acetamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(pyridin-4-ylmethyl)piperazine-1-carboxamide
N-ethyl-4-methoxy-N-(2-methylprop-2-en-1-yl)-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-[(2-methoxyphenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-ethoxy-6-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
1-ethyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1H-pyrazole-4-sulfonamide
(1R,3S)-7-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
1-[(2-fluorophenyl)methyl]-N-methyl-N-(quinolin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-3-(2-hydroxyethyl)piperazin-2-one
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
6-methyl-5-[4-(1H-pyrazol-5-yl)phenyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[3-(methylsulfanyl)phenyl]methyl}-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
methyl 5-[2-(cyclohexylmethyl)morpholin-4-yl]-5-oxopentanoate
8-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2,5-dimethyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]thiophene-3-sulfonamide
methyl 3-{[(5-methylthiophen-2-yl)formamido]methyl}-5-(quinoline-8-sulfonamido)benzoate
N-[(3-fluorophenyl)methyl]-5-(methoxymethyl)furan-2-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-[(quinazolin-4-yl)amino]pentan-1-one
3-(3,4-dimethoxyphenyl)-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
5-acetyl-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]thiophene-2-carboxamide
3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrimidin-3-yl}benzamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-amine
N-[1-(pyrazin-2-yl)piperidin-3-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[(2R,3S,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N-(propan-2-yl)propanamide
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(dimethylamino)-N-methyl-2-(3-methylphenyl)acetamide
5-acetyl-3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
6-(3-hydroxyphenyl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3aS,6aR)-5-{[2-(difluoromethoxy)phenyl]methyl}-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-5-tert-butyl-1H-pyrazole
(3S,5S)-1-benzyl-N-[(2,3-dimethoxyphenyl)methyl]-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
(4aS,7aR)-1-(pyridazine-3-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-8-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-(4-methoxyphenyl)-3-phenylpropanamide
3-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
(1S,5R)-3-[(5-methylfuran-2-yl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-butyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1,3-benzoxazole-5-carboxamide
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
2-(2H-1,3-benzodioxol-5-yl)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-[(2,3-dimethoxyphenyl)methyl]-1-(9H-purin-6-yl)piperidin-4-amine
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
N-({1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)-3,5-dimethoxybenzamide
2-(2-aminoethyl)-N-(cyclopropylmethyl)-N-(2-methoxyethyl)quinazolin-4-amine
1-({4-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]phenyl}methyl)piperidine
3-[2-(azepan-1-yl)-2-oxoethyl]-4-(2,3-dihydro-1H-inden-2-yl)piperazin-2-one
1-ethyl-4,6-dimethyl-3-(thiomorpholine-4-carbonyl)-1,2-dihydropyridin-2-one