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N-propyl-5-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}pyrimidin-2-amine
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-{[({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)amino]methyl}-1,2-dihydroquinolin-2-one
3-{[3-cyclopropyl-1-(3,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
N-[(3R,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
2-(pyridin-3-yl)-N-[3-(pyridin-3-yloxy)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl){[2-(trifluoromethyl)phenyl]methyl}amine
4-(3-methoxyphenyl)-3-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazole
methyl (2S)-2-({1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-3-phenylpropanoate
6-(2H-1,3-benzodioxol-5-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
1-(3-phenylpropyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-{[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl](propan-2-yl)amino}propanamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
N-({7-[2-(naphthalen-1-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
(1S,2R)-1-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-2,3-dihydro-1H-inden-2-ol
8-cyclobutyl-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-methyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}-3-methoxyphenol
3-ethyl-N-({7-[3-(2-methoxyphenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
(2E)-3-(1H-imidazol-4-yl)-1-{4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}prop-2-en-1-one
1-[3-(4-{[(cyclohexylmethyl)amino]methyl}-2-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
6-methyl-4-[2-methyl-4-(2-methylphenyl)-5-oxopiperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-chloro-4-[1-(2-hydroxy-2-phenylethyl)-1H-imidazol-2-yl]phenol
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl 5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-5-oxopentanoate
2-[(4-chlorophenyl)methyl]-4-{4-[(3,4-dimethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
6-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyridine-2-carbonitrile
2-(4-fluorophenoxy)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
1-[2-(4-methoxyphenyl)ethyl]-N-methyl-N-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2-ethyl-2,5-dihydro-1H-pyrrole
5-[2-(difluoromethoxy)phenyl]-1-(2-fluoroethyl)-4-phenyl-1H-imidazole
2-(2-phenyl-1H-imidazol-1-yl)-1-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}ethan-1-one
N-[(3R,5S)-1-ethyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-3,5,7-trimethyl-1H-indole-2-carboxamide
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
3-{1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyridine
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-(2,4-difluorophenoxymethyl)-1H-pyrazole
2-fluoro-6-methoxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
3-(2-ethyl-1H-imidazol-1-yl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}propan-1-one
5-[(2-acetamidoethyl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
N-ethyl-3-[2-(4-fluorophenyl)morpholin-4-yl]-N-phenylpropanamide
1-methyl-1-(2-oxo-2-{3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}ethyl)urea
5-methyl-1-[4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]pyrrolidin-2-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
7-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine