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(1R,5R)-3-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2,6-dimethylphenyl)-4-(2,5-dioxo-4-propylimidazolidin-4-yl)piperidine-1-carboxamide
N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2-phenylethyl)propanamide
3-bromo-5-(cyclohexylsulfamoyl)benzoic acid
(3R,4S)-4-cyclopropyl-1-phenylmethanesulfonylpyrrolidin-3-amine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-benzothiophene-2-carboxamide
1-(cyclopropylmethyl)-5-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-({4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
N,N-dimethyl-1-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
6-{pyrazolo[1,5-a]pyridin-7-yl}-2,4-dihydro-1H-3,1-benzoxazine-2,4-dione
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-5-methylpiperidin-2-one
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
[4-({1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-[2-(piperidin-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{[2-(2-benzamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenyl-1H-pyrazole-5-carboxamide
3-methyl-4-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3,4-dihydroquinazoline-7-carboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
2-[2-(1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)ethyl]pyridine
3,3,3-trifluoro-2-hydroxy-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}propanamide
2-[4-(1H-imidazol-4-ylmethyl)piperazin-1-yl]-1,3-benzothiazole
4-{3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]phenyl}-4H-1,2,4-triazole
3-[(4-methoxyphenyl)methyl]-4-(1-phenylethyl)-4H-1,2,4-triazole
1-ethyl-3-(2-methylpropyl)-5-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
N-(4-methylphenyl)-3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
(4S)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-1,3-oxazolidin-2-one
ethyl 4-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
3-[(4-methoxyphenyl)methyl]-4-(4-methylphenyl)-4H-1,2,4-triazole
4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
3-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
3-[(methylsulfanyl)methyl]-5-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1,2,4-oxadiazole
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-butyl-N-[(3-methylthiophen-2-yl)methyl]-4-oxoadamantane-1-carboxamide
[2-(6-aminopyridin-2-yl)phenyl]methanol
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(1H-1,2,3,4-tetrazol-5-yl)acetamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
4-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperazin-1-yl]-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(2,5-dimethylphenyl)-3-[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]propanamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-(2,4,6-trifluorophenyl)acetamide
4-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
methyl 1-methoxy-2-oxo-8-[3-(trifluoromethyl)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{[4-(aminomethyl)phenyl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-[(3R,4S)-4-(5-methylfuran-2-yl)-1-(oxane-4-carbonyl)pyrrolidin-3-yl]methanesulfonamide
2-(diethylamino)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
(2E)-3-(furan-2-yl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)prop-2-enamide
methyl 1-[(3R,5S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5-[(diphenylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylpyrimidine-5-carboxamide
(1S,5R)-6-(3-chloro-1H-indole-2-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane