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1-(2-methylpropyl)-4-(2-phenyl-1,3-thiazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(3,5-dimethylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2R,3R)-1'-[3-(dimethylcarbamoyl)propanoyl]-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(2,5-dimethylfuran-3-carbonyl)piperidine-4-carboxylate
1-{[4-(2,3-dihydro-1,4-benzodioxin-6-yloxy)-3-ethoxyphenyl]methyl}pyrrolidine
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2,5-dimethylphenyl)piperazine
2-[3-(2-oxoazepan-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclobutan-1-amine
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]amine
(3R,4R)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
ethyl 1-{[4-(ethoxycarbonyl)-1-(4-methoxyphenyl)-1H-pyrazol-5-yl]methyl}piperidine-3-carboxylate
2-(4-methyl-1H-pyrazol-1-yl)-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-fluoro-6-hydroxybenzamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)thiophene-3-carboxamide
3-cyclopropyl-5-(1-phenyl-1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazole
5-phenyl-4-{1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}-2-(trifluoromethyl)pyrimidine
3-{1-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}propan-1-ol
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
5-butyl-1-(4-chlorophenyl)-4-(3-hydroxypropanoyl)piperazin-2-one
methyl 2-methyl-2-[3-(1-methylpiperidin-2-yl)propanamido]propanoate
(3R,5S)-N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-[5-(3-cyclopropyl-1H-pyrazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-methyl-1H-1,3-benzodiazole
7-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-[(3E)-pent-3-enoyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(2-phenyl-1,3-thiazol-4-yl)methyl]amine
2-acetyl-8-{[2-(propylamino)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}-5-methoxypyridin-4-ol
2-(adamantan-1-yl)-N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
4-chloro-3-fluoro-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}benzamide
7-(3-chlorophenyl)-4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[2-({[2-(ethylsulfanyl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylacetamide
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
N-methyl-N-[3-(2-methylphenoxy)propyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
4-[3-(2,4-difluorophenyl)propanoyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S,4S)-4-amino-1-[2-(azepan-1-yl)-2-oxoacetyl]-N,N-diethylpyrrolidine-2-carboxamide
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-(1H-pyrazol-1-yl)butan-1-one
{1-[2-(4-chlorophenoxy)ethyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-hydroxy-3,5-dimethylphenyl)methyl]piperidin-3-yl}propanamide
3-chloro-N-(3-{2-methoxy-4-[(3-methylpiperidin-1-yl)methyl]phenoxy}propyl)benzamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
methyl 4-[(5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazol-3-yl)formamido]butanoate
(3S,9aR)-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-4-(1-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}ethyl)piperazine
(2R,6S)-2,6-dimethyl-4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)morpholine
(2E)-3-(4-chlorophenyl)-1-[4-(2-phenylpyrimidin-4-yl)piperidin-1-yl]prop-2-en-1-one
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-2-(trifluoromethyl)benzene-1-sulfonamide
1-methyl-5-{1-[4-(methylsulfanyl)phenyl]-1H-1,2,4-triazol-5-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione