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ethyl 4-oxo-5-phenoxy-1-(quinolin-8-yl)-1,4-dihydropyridine-3-carboxylate
(3S)-1-{1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}pyrrolidin-3-ol
4-{1-butyl-5-[(2-oxo-1,3-oxazolidin-3-yl)methyl]-1H-1,2,4-triazol-3-yl}benzamide
(3R,4R)-1-(2-chloro-4-fluorobenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
7-(1-ethyl-1H-pyrazole-3-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-({4-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)azetidin-3-ol
1-(1-methyl-1H-pyrrol-2-yl)-2-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}ethane-1,2-dione
1-(1-{[1-(oxan-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)cyclopentan-1-ol
1-cyclopropyl-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
6-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole
2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-(dimethylamino)-N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(3-methylphenyl)acetamide
1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
N,N-dimethyl-3-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
2-(2-oxo-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-[(4-chlorophenyl)(phenyl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
2-[4-(4-aminopyrimidin-2-yl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(4-fluorophenyl)-1-(1,3-thiazol-2-ylmethyl)piperidin-3-amine
{2-[(1H-imidazol-2-ylmethyl)[(5-methylthiophen-2-yl)methyl]amino]ethyl}dimethylamine
(1S,6R)-3-methyl-9-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
3-ethyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(methylamino)pyridine-4-carboxamide
2-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}-1-phenylethan-1-ol
2-{5-[(3,4-dimethoxyphenyl)methyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
N-[2-(benzyloxy)ethyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
[3-(3-phenylpropyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl]methanol
2-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
methyl 4-(5-{[3-(ethylcarbamoyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-2,4-dimethylpyridine
5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-3-(2-methylpropyl)-1H-1,2,4-triazole
N-[(3R,4R)-3-hydroxy-1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl]pyridine-4-carboxamide
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
5-{3-[3-(pyrrolidin-1-yl)propyl]-1,2,4-oxadiazol-5-yl}-1H-indole
3,4,7-trimethyl-2-[2-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1H-indole
4-(1-hydroxy-2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)phenol
(1S,2S)-2-{4-[3-(2H-1,3-benzodioxol-5-yl)propyl]piperazin-1-yl}cyclohexan-1-ol
1-[(3-fluorophenyl)methyl]-6-oxo-N-[3-(pyridin-4-yl)propyl]piperidine-3-carboxamide
8-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(4-{[4-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methanol
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
N-[1-(cyclohex-1-en-1-yl)ethyl]-1-(pyrazine-2-carbonyl)piperidin-4-amine
N-[2-(dimethylamino)ethyl]-2-{4-[(3-phenyl-1,2-oxazol-5-yl)methyl]morpholin-3-yl}acetamide
2-(2H-1,3-benzodioxol-5-yl)-1-[(3S,4S)-3-(4,4-difluoropiperidin-1-yl)-4-hydroxypyrrolidin-1-yl]ethan-1-one
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(furan-2-ylmethyl)(prop-2-en-1-yl)amine
(1R,5R)-6-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane