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1-methyl-5-[(2,2,2-trifluoro-1-phenylethoxy)methyl]-1H-1,2,4-triazole
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
1-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]urea
4-[1-(4-fluorophenyl)piperidin-4-yl]-2-(trifluoromethyl)morpholine
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]oxan-4-amine
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]-6-methoxyphenol
3,5-dimethyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
4-[2-(1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)ethyl]morpholine
3-[1-(1-benzylpiperidin-4-yl)-1H-imidazol-2-yl]phenol
1-{3-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}-N,N-dimethylpyrrolidin-3-amine
4-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-N-(pyridin-4-ylmethyl)aniline
4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
1-(carbamoylmethyl)-N-(5-methyl-2-pentanamidophenyl)piperidine-3-carboxamide
[2-propoxy-5-(quinolin-6-yl)phenyl]methanol
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-phenyl-1,2-oxazole-3-carboxamide
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(piperidin-1-yl)ethyl]acetamide
2-methoxy-1-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
1-{5-[(butylamino)methyl]-2-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)methanamine
(1-methyl-1H-imidazol-2-yl)(1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)methanol
1-[(2-chlorophenyl)methyl]-N-(1-methoxybutan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-{[1-(1-benzylpyrrolidin-3-yl)-1H-1,2,3-triazol-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
({4-ethyl-5-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-cyclohexyl-5-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}pyrimidine
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine-4-carboxamide
N-(1-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carboxamide
2-{[4-cyclopropyl-5-(1-ethyl-1H-pyrazol-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(4-fluorophenyl)-4-[1-(thiophene-2-carbonyl)piperidin-3-yl]piperazine
(3S,4S)-4-cyclopropyl-1-{1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazole-5-carbonyl}pyrrolidine-3-carboxylic acid
N-[2-(dimethylamino)ethyl]-6-(4-fluorophenyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyrimidin-2-amine
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(3-methylpyridin-4-yl)piperazin-1-yl]methyl}piperidin-2-one
methyl 5-(benzylamino)-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(4aR,7aS)-1-benzyl-4-[(2-methylpyrimidin-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-ethyl-1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-[(5-methylfuran-2-yl)methyl]urea
1-[3-(3-fluorophenyl)phenyl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-amine
3-(3-methylthiophene-2-carbonyl)-1-phenylmethanesulfonylpiperidine
4-(1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidine-4-carbonyl)morpholine
(2S,4S)-1-benzyl-N-[2-(2-fluorophenyl)ethyl]-4-{[(2,4,5-trimethoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-butyl-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-1-carboxamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(3-phenylpropyl)-1,4-diazepane
N-[(1S,2R)-2-aminocyclobutyl]-6-oxo-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraene-12-carboxamide
{[1-({1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methyl}urea
5,6-dimethyl-2-{[4-(pentan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-1,3-benzodiazole
4-(3-cyclohexylpyrrolidine-1-carbonyl)-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole
3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]amine
ethyl 2-{1-[2-(2H-1,3-benzodioxol-5-yloxy)propanamido]cyclohexyl}acetate
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(4-methoxyphenyl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine