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(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(3-phenylpropanoyl)-decahydro-1,6-naphthyridin-2-one
N-{1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-(1-{2-oxo-2-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl}-1H-pyrazol-4-yl)thiophene-3-carboxamide
(5S,9aS,9bS)-5-[4-methoxy-3-(methoxymethyl)phenyl]-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-3,5-dimethoxybenzamide
9-oxo-N-propyl-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecane-2-carboxamide
(2S,4R)-1-(4-acetylbenzenesulfonyl)-4-amino-N,N-diethylpyrrolidine-2-carboxamide
1-(3,5-dimethylphenyl)-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
1-[(2-chlorophenyl)methyl]-N-ethyl-N-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-4-methoxyphenol
N-[1-(2-phenylethyl)piperidin-3-yl]quinoxaline-6-carboxamide
[(2S,4R)-4-(dimethylamino)-1-[1-(2-methylbenzoyl)piperidine-4-carbonyl]pyrrolidin-2-yl]methanol
6-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzothiazol-2-one
(1S,5R)-6-benzyl-3-(5-methyl-1H-indazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-tert-butyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide
4-[2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-2-yl)ethyl]phenol
3-(3-fluorophenyl)-N-methyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-{2-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}piperidin-2-one
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-(2,4,5-trifluorobenzoyl)piperidin-4-ol
2-oxo-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-oxaspiro[4.4]nonane-4-carboxamide
N-(3-cyanophenyl)-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
8-methyl-2-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
N-(1H-indazol-7-yl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carboxamide
N-{3-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-N-methylaniline
1-[(4aR,8aS)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridin-1-yl]-2-(2H-1,3-benzodioxol-5-yl)ethan-1-one
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyrimidin-4-yl)ethyl]amine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}(methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
1-[3-(3-{4-azaspiro[2.5]octan-4-ylmethyl}phenoxy)-2-hydroxypropyl]piperidin-4-ol
3-[2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethyl]-1H-indole
N-methyl-4-oxo-1-(3-phenylpropyl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-(furan-2-ylmethyl)-4-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidine
3-(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-4-(3-methylbutyl)piperazin-2-one
1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)cyclopropane-1-carboxamide
1-(cyclohexylmethyl)-6-oxo-N-[3-(pyridin-2-yl)propyl]piperidine-3-carboxamide
2-{[2-(diethylamino)ethyl]amino}-N-(2-fluoro-5-methylphenyl)acetamide
N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-methyl-5-{[(6-methylhept-5-en-2-yl)amino]methyl}pyrrolidin-2-one
4-amino-1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}butan-1-one
4-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-N-methylpyridin-2-amine
2-(2,6-dimethoxypyridin-3-yl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
3-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1H-indazole
1-(3-chloro-4-fluorophenyl)-5-(cyclopropylmethyl)-3-methyl-1H-1,2,4-triazole
3-[(3R,4S)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-[(3-methoxyphenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide