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N-tert-butyl-4-{3-[(2-phenylethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
1-[1-(3-fluorobenzoyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
2-(2-methoxyphenyl)-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]acetamide
2-cyclopropyl-N-[3-(4-methylpiperazin-1-yl)butyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]acetamide
5-(1-butyl-1H-1,2,4-triazol-5-yl)-N-(propan-2-yl)pyrimidin-2-amine
5-{imidazo[1,2-a]pyrimidin-2-yl}-3-(2-methoxyphenyl)-1,2,4-oxadiazole
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
3-(4-hydroxyphenyl)-1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-2-phenylpropan-1-one
4-(pyridin-2-yl)-N-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]acetamide
1-(1H-imidazol-2-ylmethyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(1H-indazol-6-yl)-4-[2-(methylsulfanyl)pyridine-3-carbonyl]piperazin-2-one
2-methoxy-N-[(2R,3R)-2-methoxy-1'-(4-methyl-1,3-oxazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
[(3-{[1-(4-methoxybenzoyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(quinolin-5-ylmethyl)amine
N-[2-(4-cyclopentylmorpholin-2-yl)ethyl]-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
1-ethyl-N-[3-(1H-imidazol-1-yl)butyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(2-hydroxyethyl)-N-methyl-1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(furan-2-ylmethyl)piperidine
[(3-fluorophenyl)methyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
N'-(2-ethoxyphenyl)-N-[(2-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)propanediamide
2-methyl-4-{3-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]phenyl}but-3-yn-2-ol
3-[6-amino-5-cyano-4-(furan-3-yl)pyridin-2-yl]benzoic acid
(1S,5R)-3-(9H-purin-6-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[5-(2,3,4-trimethoxyphenyl)pyridin-2-yl]methanesulfonamide
5-(2,4-dimethoxyphenyl)-1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
N,N-dimethyl-5-{[(3-methylphenyl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-{[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(butan-2-yl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
3-chloro-5-(4-phenylazepane-1-carbonyl)-1,2-dihydropyridin-2-one
4-{4-[(2,3-dihydro-1-benzofuran-3-yl)amino]piperidin-1-yl}-N,N,6-trimethylpyrimidin-2-amine
4-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1H-imidazole-5-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]acetamide
5-(3-fluorophenoxymethyl)-N-(5-methylhexan-2-yl)-1H-pyrazole-3-carboxamide
4-{7-fluoro-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carbonyl}-1,3-dimethylpiperazin-2-one
4-[1-(2,3,4-trimethoxybenzoyl)piperidin-3-yl]morpholine
2-phenyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}imidazo[1,2-a]pyridine-6-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(piperidin-1-yl)ethyl]acetamide
methyl 1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-4-carbonyl]piperidine-4-carboxylate
4-cyclobutaneamido-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
4-[(dimethylamino)methyl]-1-(4-phenoxybutyl)azepan-4-ol
methyl 3-{[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}propanoate
N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[1-(thiophen-2-yl)ethyl]benzamide
N-{1-[(3-methylphenyl)methyl]cyclopropyl}spiro[2.2]pentane-1-carboxamide
[(3-{[1-(2,5-dimethoxybenzoyl)piperidin-4-yl]oxy}-4-methoxyphenyl)methyl](methyl)(propan-2-yl)amine
N-(3-chloro-4-fluorophenyl)-3-[1-(thian-4-yl)piperidin-4-yl]propanamide
5-methoxy-3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
2-(1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-1,3-benzoxazole
1-ethyl-4,6-dimethyl-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[2-({4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine