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3-{[(2R)-2-methylpiperazin-1-yl]sulfonyl}-N-(1,2-oxazol-3-ylmethyl)benzamide
N-[3-(3-methoxyphenyl)phenyl]-1-(1H-pyrrole-3-carbonyl)piperidine-4-carboxamide
1-cyclopropyl-3-{2-[2-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N-(1H-imidazol-4-ylmethyl)-N-[(3-methylthiophen-2-yl)methyl]cyclopentanamine
N-[(3R,4S)-1-(furan-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
1-(2,4-dimethylphenoxy)-3-[(4,4,4-trifluorobutan-2-yl)amino]propan-2-ol
2-{4-[(6-fluoroquinolin-2-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
(1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-[4-(4-methoxyphenyl)butan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(4-formylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-(2-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
8-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2,4-difluorophenyl)-5-[(4-fluoro-3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-2-methylpropanoic acid
2-phenoxy-N-[2-(7-{[4-(pyrrolidin-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
1-(1-acetylpiperidin-4-yl)-N-benzylpiperidine-3-carboxamide
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
1-{4-[(1-methoxybutan-2-yl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-ethylpiperidine
[(4aS,8aR)-6-(pyridine-3-sulfonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N,3-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}furan-2-carboxamide
2-ethyl-4-{4-phenyl-1-[3-(pyrrolidin-1-yl)propyl]-1H-imidazol-5-yl}pyrimidine
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N,N-dimethylpyridine-3-carboxamide
3-({cyclopropyl[(3-hydroxyphenyl)methyl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1-methyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}-1,2-oxazol-5-yl)methyl]-N-methylacetamide
(3aS,6aS)-2-[(3-hydroxyphenyl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[(4-methylphenyl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
4-[(4-chloro-3-fluorophenyl)methyl]-1,4-oxazepan-5-one
5-ethyl-N-[3-(methylsulfanyl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-{[1-(dimethylamino)butan-2-yl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-(4-hydroxyphenyl)-N-(3-hydroxypropyl)-N-[(4-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
1-[1'-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[(2-fluoro-3-methoxyphenyl)methyl]-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)methylamine
3-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-[2-(morpholin-4-ylmethyl)phenyl]urea
6-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2,4-dimethylpyridine-3-carbonitrile
1-[(2S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
(4aR,8aR)-2-(2,1,3-benzoxadiazol-4-ylmethyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
1-(2-methylpentyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
3-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
N-(3-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)carbamoyl]methoxy}phenyl)propanamide
1-(3,4-dichlorobenzoyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
N6-cyclopropyl-N4-methyl-N4-[2-(pyridin-2-yl)ethyl]pyrimidine-2,4,6-triamine
2-(trifluoromethyl)-4-(2,3,4-trimethoxybenzoyl)morpholine
2-[4-(1-ethoxyethyl)phenyl]pyridine-3-carbonitrile
(2S,3S)-2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]-3-methylpentanamide
methyl 9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-3-{[4-(propan-2-yl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate