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1-{3-[4-(4-fluorophenoxy)piperidin-1-yl]-3-oxopropyl}azepan-2-one
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(thiophen-2-yl)propan-1-one
4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1λ6-thiane-1,1-dione
2-hydroxy-N-methyl-N-(quinolin-5-ylmethyl)pyridine-3-carboxamide
4-(1,2,4-oxadiazol-3-yl)-1-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)piperidine
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-2-one
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-3,6,7-trimethyl-1-benzofuran-2-carboxamide
6-(1-benzothiophen-3-yl)-2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)pyridine-3-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-fluorophenyl)ethyl]acetamide
N-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-(thiophen-3-yl)acetamide
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
1-methyl-4-[(6-methylquinolin-5-yl)methyl]piperazine-2-carboxylic acid
3-[(2,5-dimethylphenyl)[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl]pyridine
4-({2-[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}methyl)-1-ethylpyrrolidin-2-one
(3R,4R)-1-[(2-ethoxyphenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4H-chromen-4-one
2-{1-[1-(thiophene-2-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-(thiophen-2-yl)pyrimidin-4-ol
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
2-(3-fluorophenoxymethyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
ethyl 4-[(2S,4R)-4-(dimethylamino)-2-(methoxycarbonyl)pyrrolidin-1-yl]piperidine-1-carboxylate
7-(pyrazine-2-carbonyl)-N-(thiolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-methyl-N-{1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-2-phenylethyl}-2-(1H-pyrazol-1-yl)acetamide
4-(pyrazin-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(3S,9aR)-3-benzyl-2-methyl-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}cyclopropanesulfonamide
[(3R,4R)-1-(5-chloro-2-fluorobenzoyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
(1S,5R)-6-cycloheptanecarbonyl-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[(3-methyloxetan-3-yl)methyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-{3-[2-(3,4,5-trimethoxyphenyl)-1H-imidazol-1-yl]phenyl}-1H-1,2,3,4-tetrazole
methyl 1-[(4-{[(4-methylphenyl)methyl]amino}quinazolin-2-yl)methyl]piperidine-2-carboxylate
(2R,3R)-3-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[4-(hexyloxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(2S,4R)-4-(2H-1,3-benzodioxole-5-amido)-1-(1H-imidazol-2-ylmethyl)-N-methylpyrrolidine-2-carboxamide
3-(2,6-dimethylpyridin-3-yl)-1-[3-(4-methylbenzenesulfonamido)propyl]urea
ethyl 2-(1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
6-(methoxymethyl)-N,1-dimethyl-N-[2-(phenylsulfanyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
4-(1-{[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]amino}ethyl)hepta-1,6-dien-4-ol
5-[1-(methoxymethyl)cyclopropyl]-3-[2-(methylsulfanyl)ethyl]-1-propyl-1H-1,2,4-triazole
1-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-3-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
2-[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-4-carboxamide
3-[6-(2-methoxyphenyl)pyridazin-3-yl]benzonitrile
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methyl-1,2,5-oxadiazole-3-carboxamide
6-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}pyridine-2-carboxylic acid