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5-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(3,4-dimethoxyphenyl)methyl]-N-(2-methoxyethyl)-N-(propan-2-yl)-1,3-benzoxazole-6-carboxamide
1-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-3-carboxamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,2,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(4-methoxyphenoxymethyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
1'-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-(hydroxymethyl)pyridine-2-carboxamide
1-methyl-N-{[8-(quinolin-8-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-pyrazole-3-carboxamide
N-(3-methoxypropyl)-5,6-dimethyl-N-{[2-(3-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2,5-dimethylphenyl)-3-methyl-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2-hydroxy-6-methyl-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
2-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
1-[(2-methoxyphenyl)methyl]-N-methyl-N-[(4-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
5-(1H-pyrazol-3-yl)-2-(1H-pyrrol-1-yl)pyridine
3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N2,N2-dimethyl-N4-[2-(pyridin-3-yloxy)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-{1-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-chlorophenyl)-4-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}piperazin-2-one
2-(ethylamino)-N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]pyrimidine-5-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(3-ethynylbenzoyl)piperidin-3-yl]propanamide
4-(4-cyclopentylpyrimidin-2-yl)-N-cyclopropylpiperazine-2-carboxamide
2-(5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,2,4-oxadiazol-3-yl)pyridine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-5,6-dimethylpyridine-3-carboxamide
4-({2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-N-(1,3-thiazol-2-yl)benzamide
[1-(4-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methanol
N,N-dimethyl-5-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyrimidin-2-amine
methyl 5-{[(3-ethoxy-4-methoxyphenyl)methyl]amino}-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]-1-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}piperidine
6-[4-(propan-2-yl)phenyl]pyridine-3-carboxamide
3-tert-butyl-1-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}urea
1-(6-ethyl-2-methylquinoline-4-carbonyl)-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
1-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}piperidine
3-(4-methoxyphenyl)-N-(oxan-4-yl)-1H-pyrazole-5-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-1-phenylcyclopropane-1-carboxamide
5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
{1-[(2-chloro-4-fluorophenyl)methyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
N-(4-chlorophenyl)-3-[1-(5-phenylpentanoyl)piperidin-3-yl]propanamide
3-({[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
2-ethoxy-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
8-[2-(benzenesulfonyl)ethyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea