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3-(aminomethyl)-N-(4-phenoxyphenyl)piperidine-1-carboxamide
(2E)-N-{2-[4-(1H-pyrazol-5-yl)phenyl]phenyl}but-2-enamide
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propane-1-sulfonamide
N-[(3R,4S)-1-(4,6-dimethylpyridine-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-benzyl-N3-cyclopropyl-N5-[(2,6-difluorophenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-(4-ethoxy-3-methylphenyl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}butan-1-one
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-1-methylpiperidine-4-carboxamide
(1R,3S)-3-ethoxy-7-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
N-ethyl-2-(1H-imidazol-1-yl)-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)acetamide
5-(2-methoxyacetamido)-1-methyl-N-(2-methylbutyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
2-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}quinoline
N-methyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(1,4-dioxan-2-ylmethyl)-N-methylacetamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]propanamide
4-(1H-pyrazol-4-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}butanamide
5-oxo-1-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-3-carboxylic acid
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-(quinolin-8-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
methyl 7-oxo-9-(pyridin-3-ylmethoxy)-3-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(1H-indol-3-yl)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
1-ethyl-3-(morpholine-4-carbonyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methyl-5-[3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(3-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
1-cyclohexyl-3-(2,4-dimethoxybenzoyl)piperidine
2-(1,4-dimethylpiperazin-2-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)acetamide
4-methyl-2-{1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-yl}-1H-1,3-benzodiazole
2-[(4-chlorophenyl)methyl]-8-(4-methoxypyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}benzamide
1-benzyl-N3-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-(4-fluorophenyl)-2-methyl-4-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-3-yl}pyrimidine
3-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(1H-1,3-benzodiazol-1-yl)-1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
4-[7-(2-chloropyridine-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
N-[2-(dimethylamino)ethyl]-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-ethyl-1-[2-(4-fluorophenyl)azetidin-1-yl]pentan-1-one
N-[(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-5-oxopyrrolidine-2-carboxamide
N-ethyl-3-[4-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-cyclopropyl-1-(2-methoxyphenyl)-5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazole
(1S,5R)-3-[4-(5-methylfuran-2-yl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(5-fluoro-1H-indol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-amino-6-(2,2-dimethyloxan-4-yl)-4-(1-ethyl-1H-pyrazol-4-yl)-5-methylpyridine-3-carbonitrile
1-cyclopentyl-4-{3-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenoxy}piperidine
N-({1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(1-phenyl-1H-imidazol-4-yl)benzamide
4-[4-(1-hydroxy-2-methylpropyl)piperidin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
1-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one