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(5S,9aS,9bS)-5-[(E)-2-(4-fluorophenyl)ethenyl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
4-cyclobutanecarbonyl-7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrazolo[1,5-a]pyridine-7-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-({1-[(2E)-2-methylpent-2-en-1-yl]pyrrolidin-3-yl}methyl)urea
2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-ylmethyl}benzonitrile
5-[(3,4-difluorophenyl)methyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
2-methoxy-1-(4-{4-[2-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(6-methylpyridin-2-yl)methyl]amino}pyrrolidine-2-carboxamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-4-carboxamide
N,N-diethyl-1-[(4-{[4-(2-hydroxyethoxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidine-3-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[(3-ethoxy-4-methoxyphenyl)methyl]-N-methylacetamide
1-ethyl-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)benzoic acid
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]but-3-en-1-one
4-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
4-[4-(2-methylphenoxy)piperidin-1-yl]-4-oxobutane-1-sulfonamide
1-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}piperidine-3-carboxamide
N-[(3S,5S)-1-acetyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-(3-chlorophenyl)-4-[2-(2-ethylpiperidin-1-yl)acetyl]piperazin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1-{7-[2-(3-fluorophenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperazine
N-[(3R,4S)-1-cyclopentyl-4-cyclopropylpyrrolidin-3-yl]-4-(1H-imidazol-1-yl)butanamide
methyl (1R,3S,3aR,6aS)-3-(3-ethoxy-2-hydroxyphenyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-[(3-fluorophenyl)methyl]-4-{4-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(5-{1-[(4-methanesulfonylphenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
N-(3,5-dimethylphenyl)-6-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-[3-(furan-2-yl)benzoyl]-4-(4-methoxybenzoyl)piperazine
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
6-(morpholin-4-yl)-N4-(oxan-4-ylmethyl)pyrimidine-2,4-diamine
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-[(2,3-dimethoxyphenyl)methyl]-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
4-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-N-(2-hydroxyethyl)pyridine-2-carboxamide
5-[4-(4-tert-butylphenyl)-4-oxobutyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-{[1-(methoxymethyl)cyclopentyl]methyl}-2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H-imidazole
2-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(2-methoxyphenoxy)-N-methylacetamide
3-{4-[(8-methoxy-2H-chromen-3-yl)methyl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
methyl 4-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)thiophene-2-carboxylate
3-(5-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-yl}-1,2,4-oxadiazol-3-yl)pyridazine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
N-[(1-ethyl-1H-indazol-3-yl)methyl]-8-fluoroquinoline-2-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(2,5-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide