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N-[(1R,3R)-3-aminocyclopentyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
5-benzamido-N-butyl-1-cyclopentyl-N-methyl-1H-1,3-benzodiazole-7-carboxamide
(2R,3R)-3-amino-1'-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-4-(1H-imidazol-2-yl)piperidine
3-{[4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]sulfonyl}pyridine
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-propylpentanamide
2-methyl-6-[1-(1-methylpiperidin-4-yl)-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]pyridine
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
2-methyl-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-3-phenylcycloprop-2-ene-1-carboxamide
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-{[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
2-methyl-4-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-4,5,6,7-tetrahydro-1,3-benzothiazole
N-methyl-4-{3-methyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}-1,3-thiazol-2-amine
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(morpholine-4-carbonyl)piperidin-1-yl]ethan-1-one
ethyl 1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine-3-carboxylate
3-(2-{6-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-methoxyphenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)acetamide
N-[(3R,4S)-1-(3-cyano-4,6-dimethylpyridin-2-yl)-4-propylpyrrolidin-3-yl]-3-methoxypropanamide
(1S,5R)-6-[1-(4-methylphenyl)cyclopropanecarbonyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(5-methylthiophene-3-carbonyl)pyrrolidin-3-yl]methanol
N-{3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}acetamide
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
3-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
3-(3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-3-oxopropyl)-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{[(5-ethylpyridin-2-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}propan-1-ol
1-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
N-{4-[3-(pyridin-3-yl)propanamido]phenyl}pentanamide
{[1-(2H-1,3-benzodioxol-5-yl)-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl]methyl}urea
(3S,5R)-1-(cyclopropylmethyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
5-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
2-methoxy-5-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}benzoic acid
1-methyl-2-(5-{1-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)-1H-1,3-benzodiazole
3-{[(2-aminopyridin-3-yl)methyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
7-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-oxa-7-azaspiro[4.5]decane
[2,2-dimethyl-3-(morpholin-4-yl)propyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
(2R)-2-amino-N-[(2-methylphenyl)methyl]-2-phenyl-N-(prop-2-en-1-yl)acetamide
8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-{[2-(trifluoromethoxy)phenyl]methyl}oxane-2-carboxamide
1-[(1-{6-[(pyrrolidin-3-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(3R,4R)-3-cyclobutyl-4-methyl-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyrrolidin-3-ol
3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}urea