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2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-4-phenoxybutanamide
3-methyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
N-(3-ethoxypropyl)-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
8-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(morpholin-2-yl)acetamide
(2S)-N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-2-(methoxymethyl)pyrrolidine-1-carboxamide
2-ethyl-4-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazole-5-carboxamide
8-(naphthalen-1-ylmethyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
ethyl 1-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carbonyl]piperidine-2-carboxylate
1-(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
4-[5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-pyrazol-3-yl]phenol
4-(2-{[2-(pyridin-4-ylsulfanyl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzamide
8-(1,3-benzothiazol-2-ylmethyl)-1-benzyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 3-(2-methylpropyl)-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3aS,6aR)-5-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-({7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
(3S,4S)-1-(6-aminopyridine-3-carbonyl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
1-{2-[(4-methoxy-2-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-2-methylpropan-1-one
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[2-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-yl]methanol
2-[(4aR,7aS)-6,6-dioxo-4-(3,3,4,4-tetrafluorobutyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-methyl-7-(5-propyl-1,3,4-oxadiazol-2-yl)-2,7-diazaspiro[4.5]decane
(3R,4S)-4-cyclopropyl-1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-amine
3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-N-(1H-imidazol-2-ylmethyl)piperidin-4-amine
N-benzyl-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-N-methylpiperidin-3-amine
6-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-2-carboxylic acid
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
5-[2-(azepan-1-yl)-2-oxoacetyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]acetic acid
4-[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidine-3-carbonyl]morpholine
N-benzyl-N-(2-hydroxyethyl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
3-{[(1-ethylcyclopropyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
4-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}quinoline
1-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}but-3-en-1-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-1H-pyrazole-3-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1-methylpiperidine-3-carboxamide
1,4-bis(pyrimidin-2-yl)-1,4-diazepane-6-carboxylic acid
6-(1-acetylpiperidine-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-[2-(methylsulfanyl)ethyl]piperazine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(furan-2-yl)ethyl]acetamide
5-[(3,4-dimethoxyphenyl)methyl]-2-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-(morpholin-4-ylmethyl)-N-{[2-(trifluoromethyl)phenyl]methyl}furan-3-carboxamide
3,7-dimethyl-11-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-3,7,11-triazaspiro[5.6]dodecane
methyl(1-{1-[4-(morpholin-4-yl)benzoyl]piperidin-4-yl}-2-phenylethyl)(pyridin-4-ylmethyl)amine
2-(3-fluorophenoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
(3S,4R)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine