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N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
3-(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-N-cyclopropylpropanamide
4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}thiomorpholine
methyl 3-(3-ethynylbenzoyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-ethyl-N,4-dimethyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,3-oxazole-5-carboxamide
1,5-dimethyl-N-[2-(4-methylmorpholin-2-yl)ethyl]-1H-indazole-3-carboxamide
ethyl 2-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}amino)propanoate
2-(2-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenyl)-6-(oxolan-3-yl)-3,4-dihydropyrimidin-4-one
methyl 7-oxo-9-(pyridin-2-ylmethoxy)-3-[4-(thiophen-2-yl)butanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(propan-2-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}piperidine-4-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
N-methyl-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-ethyl-1,2-oxazole-3-carboxamide
ethyl 4-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]piperidine-1-carboxylate
N-[(3R,4S)-1-[(3,5-dimethoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxyacetamide
6-(2-chlorophenyl)-N-[2-(dimethylamino)butyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-chloro-N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-fluorobenzamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
ethyl 1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1-benzofuran-5-carboxamide
6-{3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
4-(4-chlorophenyl)-1-{[2-hydroxy-5-(pyridin-3-yl)phenyl]methyl}piperidin-4-ol
(4aR,7aS)-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-N-cyclohexyl-N-methylpyridine-2-carboxamide
2,3-dimethyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1H-indole-5-carboxamide
1-[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
methyl 2-{[(5-fluoro-2-methoxyphenyl)methyl]amino}pyridine-4-carboxylate
2-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}quinolin-4-ol
5-[3-(3-methoxyphenoxy)propyl]pyridine-3-carboxamide
ethyl 4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine-1-carboxylate
2-(cyclopropylmethyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2-methoxyethan-1-one
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(pyridin-2-ylmethyl)amine
N-{3-[methyl(phenyl)amino]propyl}-2,7-dioxo-1,3-diazepane-4-carboxamide
N-{2-[3-cyclopropyl-1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]ethyl}-4-methylbenzamide
{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amine
(1R,3S,5S)-8-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
(4aS,8aR)-6-(1H-imidazol-4-ylmethyl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperazine
methyl 5-(cycloheptylamino)-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(2-hydroxy-3-{4-methoxy-2-[(4-methylpiperazin-1-yl)methyl]phenoxy}propyl)piperidin-4-ol
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-(1H-pyrazol-4-yl)benzamide
6-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}quinazolin-4-amine
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-cyclopropylpropan-1-one
1-[(2,4-difluorophenyl)methyl]-5-[4-(diphenylmethyl)piperazin-1-yl]azepan-2-one
N,N-dimethyl-7-(oxolane-2-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(4-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}phenyl)methanol
(5S)-5-({[(2-methyl-1-benzothiophen-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)pyrrolidin-2-one
N-(furan-2-ylmethyl)-5-{1-[2-(1H-imidazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-ethyl-N-methylpyrazolo[1,5-a]pyrimidin-7-amine