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3-{1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-phenyl-1H-imidazol-5-yl}pyridine
5-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,4-dimethylpyridine
2-(4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
7-fluoro-3-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1-benzofuran-2-carboxamide
N-({7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
2-{9-[(3-hydroxy-4-methoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
(1S,4R)-2-{[3-(trifluoromethyl)phenyl]methyl}-2-azabicyclo[2.2.1]heptan-3-one
5-ethyl-N,2-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-4-amine
N3-(1-benzothiophen-2-ylmethyl)-1-cyclopentyl-N5,N5-diethyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(adamantan-2-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
2-[(2-methoxyethyl)(propyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(4-fluoro-2-methoxyphenyl)-2-[4-(3-fluorophenoxy)piperidin-1-yl]acetic acid
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperidin-4-ol
1-cyclopropanecarbonyl-N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]piperidine-4-carboxamide
5-(methoxymethyl)-N-({7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
5-methoxy-2-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1H-indole
1-[(3-methylthiophen-2-yl)methyl]-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[(3-fluorophenyl)methyl]acetamide
6-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(4-methylpiperidin-1-yl)propan-1-one
2-{3-oxo-9-[3-(pyridin-3-yl)propyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
2-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}morpholin-3-yl)acetic acid
1-[(4-methyl-5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-{[(3-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-cyclohexylpiperidine
1-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-1,4-diazepane
{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
(4aR,8aS)-6-[(2,5-dimethylphenyl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
{1-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]piperidin-2-yl}methanol
6-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-{[4-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}quinolin-7-ol
1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-[5-(2-chlorobenzoyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
3-({[2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
5-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrazine-2-carboxamide
4-[(3,4-dimethoxyphenyl)methyl]-7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(3-hydroxy-3-methylbutyl)-N-(3-hydroxy-3-phenylpropyl)-N-methylbenzamide
8-(2,3-dihydroxypropyl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
3-{imidazo[1,2-a]pyridin-2-yl}-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,2,4-oxadiazole
4-[(2S)-2-(piperidine-1-carbonyl)pyrrolidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[(2,6-dimethoxyphenyl)methyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-methoxy-7-(4-methoxyphenyl)-4-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[2-(1H-imidazol-4-yl)ethyl]-9-(5-methylthiophene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-5-(methoxymethyl)furan-2-carboxamide
1-[(2-fluorophenyl)methyl]-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-6-oxopiperidine-3-carboxamide
4-(2,4-dimethoxypyrimidin-5-yl)benzamide
3-[(tert-butylamino)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one