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6-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyridine-3-carboxylic acid
N-ethyl-1-{2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carbonyl}pyrrolidine-3-carboxamide
1-(2-methylpropyl)-4-[4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-diazepane
2-(4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
2-(3-chloro-4-methoxyphenyl)-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-{[1-(morpholin-4-yl)cycloheptyl]methyl}pyrrolidin-2-one
N-(2-phenylethyl)-4-[(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)oxy]benzamide
2-(benzylsulfanyl)-N4-[2-(pyridin-2-yl)ethyl]pyrimidine-4,6-diamine
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-(morpholin-4-yl)-2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-4-(1H-1,2,4-triazol-5-yl)benzamide
N-(1-cycloheptylpiperidin-3-yl)-1,5-dimethyl-1H-pyrazole-4-sulfonamide
7-(cyclohexylmethyl)-2-cyclopentanecarbonyl-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-3-(1-{[1-(propan-2-yl)-1H-indol-3-yl]methyl}piperidin-3-yl)propanamide
4-[2-(6-fluoro-2-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrazol-1-yl)propan-1-one
3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)urea
(2S,4S)-4-amino-N-methyl-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
2-[3-({[(2-fluorophenyl)methyl](2-methoxyethyl)carbamoyl}amino)phenyl]-N-methylacetamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(6-oxo-1,6-dihydropyridazin-3-yl)propanamide
6-(2-methoxyphenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2E)-1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-2-methylbut-2-en-1-one
1-methyl-5-({2-[4-(pyridin-2-yl)phenyl]-1H-imidazol-1-yl}methyl)pyrrolidin-2-one
2,3,6-trimethyl-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]quinoline
1-cyclohexyl-3-(cyclopropylmethyl)-N-(2-methoxy-2-methylpropyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-(5-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[2-(dimethylamino)benzoyl]-3-ethylpiperidine-3-carboxylic acid
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
3-methyl-4-[5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]pyridine
1-[2-(1H-pyrazol-1-yl)ethyl]-4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazole
1,9-dimethyl-10-oxo-N-(thiophen-2-ylmethyl)-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(4aS,8aR)-2-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-decahydroisoquinoline
7-(cyclopropylmethyl)-2-(7-methoxy-4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decane
1-ethyl-N-[3-(3-methylphenyl)propyl]-5-oxopyrrolidine-3-carboxamide
5-amino-N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-5-propyl-1,2-oxazole-3-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
5-(3-fluorophenyl)-3-[4-(thiomorpholin-4-yl)piperidin-1-yl]-1,2,4-triazine
5-(azocane-1-carbonyl)-2-(3-methylphenyl)pyrimidin-4-ol
1-({1-[2-(2,4-dioxoimidazolidin-1-yl)acetyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
methyl[(4-methyl-1H-imidazol-2-yl)methyl][2-(2-methylphenyl)ethyl]amine
3-(5-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-methyl-N-(1-{[methyl(oxan-2-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)furan-3-carboxamide
2-cyclopropyl-4-{4-[4-(hydroxydiphenylmethyl)piperidine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4,4-difluoropiperidine
2-[(3-methoxyphenyl)methyl]-4-(thian-4-yl)morpholine
N-[4-({4-[4-(2-methylpropyl)-2,5-dioxo-1-[2-(thiophen-2-yl)ethyl]imidazolidin-4-yl]piperidin-1-yl}methyl)phenyl]acetamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide