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(3aS,7aR)-5-methyl-2-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
N-(1,3-dihydro-2-benzofuran-5-yl)-2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carboxamide
4-(aminomethyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-(3-methoxypropyl)-8-(quinolin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[2-(2-hydroxyethoxy)ethyl]-2-(4-propanoylphenoxy)acetamide
2-{4-[(2,4-dimethoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-(1-benzothiophen-2-ylmethyl)-7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(4-methoxyphenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
1-(1-cyclopentanecarbonylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
3-[2-amino-4-methyl-6-({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amino)pyrimidin-5-yl]propanoic acid
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(3-methanesulfonamido-4-methoxyphenyl)urea
[3-(3-methylbut-2-en-1-yl)-1-[2-(pyridin-2-yl)ethyl]piperidin-3-yl]methanol
1-[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
(2E)-3-(3-fluorophenyl)-1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]prop-2-en-1-one
8-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(3-chlorophenyl)-4-[(3-{2-[1-(furan-2-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
2-{4-[(1,1-dioxo-1λ6-thian-3-yl)methyl]phenoxy}-N-methylacetamide
4-{4-[(1S,3R,3aR,6aS)-3-ethyl-3-(hydroxymethyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]phenyl}but-3-yn-1-ol
methyl[1-(1,2-oxazol-3-yl)ethyl]{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(thiophen-2-ylmethyl)amine
(2S,4R)-N-ethyl-4-[3-(5-methyl-1H-pyrazol-1-yl)propanamido]-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxamide
1-(4-{2-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-4-methoxyphenoxy}piperidin-1-yl)ethan-1-one
(1S,5R)-6-(cyclobutylmethyl)-3-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{[1-(3-cyano-4,6-dimethylpyridin-2-yl)pyrrolidin-3-yl]methyl}benzamide
4-(5-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
N-(1-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)pyridin-2-amine
6-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}quinoline
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
7-acetamido-2-(2-methoxyphenyl)-1-methyl-N-(2-phenylpropyl)-1H-1,3-benzodiazole-5-carboxamide
1-[3-(3-methoxypropyl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-5-methoxybenzamide
1-(2-chloro-5-sulfamoylphenyl)-3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]urea
3-[(3-hydroxy-4-methoxyphenyl)methyl]-9-methoxy-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-[(4-chlorophenyl)methyl]-5-{3-oxo-3-[4-(quinazolin-2-yl)piperazin-1-yl]propyl}pyrrolidin-2-one
4-(oxolane-2-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
2-[5-(5-phenyl-1,2,4-oxadiazol-3-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
4-(quinolin-2-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(1,4-dioxan-2-ylmethyl)-3-methoxy-N-methyl-4-[(1-methylpiperidin-4-yl)oxy]benzamide
3-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
1-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
N-[(2R,3R)-1'-[(2,4-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
2-{3-[3-(3-methylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}pyridine
5-{1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-[4-(3-methoxypropyl)piperazine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-cyclopropyl-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-3-phenyl-1H-pyrazole-5-carboxamide
2-hydroxy-1-[1-(hydroxymethyl)-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one