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2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
4-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-2-methyl-5-(propan-2-yl)pyrimidine
2-({[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amino}methyl)-6-methylpyridin-3-ol
[(2-chloro-5-fluorophenyl)methyl](ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
3-(1-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4-(2-methoxyethyl)piperidine-4-carboxylate
(1S,2S)-2-(4-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperazin-1-yl)cyclohexan-1-ol
3-[(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
2-[4-(4-{[(3-methylthiophen-2-yl)methyl]amino}benzoyl)morpholin-3-yl]acetic acid
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
2-amino-6-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-methoxy-5-({[(2-methylphenyl)methyl](prop-2-en-1-yl)amino}methyl)benzoic acid
N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-4-(2-oxopyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
N-(1H-1,2,4-triazol-5-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
7-(cyclobutylmethyl)-2-(pyridin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[(4-{[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(2-fluorophenyl)piperazine
2-(adamantan-1-yl)-N-(2-hydroxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-benzyl-2-[1-cyclopentyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
1-(naphthalen-2-yl)-4-(oxolan-3-ylmethyl)piperazine
4-[(dimethylamino)methyl]-1-(3-methyl-1H-pyrazole-5-carbonyl)azepan-4-ol
(4aS,8aR)-1-(3-aminopropyl)-6-{imidazo[1,2-a]pyridine-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
5-methyl-3-(4-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)-1,2,4-oxadiazole
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-ol
7-cyclohexyl-2-[2-(1H-imidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[1-(pyrazin-2-yl)piperidin-4-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N'-[2-(propan-2-yl)phenyl]-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}butanediamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}pyridine-2,4-diol
(3S,4S)-4-(dimethylamino)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
N-(3-fluorophenyl)-2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}-2-oxoacetamide
1-[1-(2,5-dimethoxyphenyl)ethyl]-2-(propan-2-yl)-1H-imidazole
[(3R,4S)-1-[(4-chlorophenyl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-ethyl-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-(oxolan-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
1-butyl-4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
methyl 4-(2-fluoro-5-methoxyphenyl)-1H-pyrrole-2-carboxylate
(2-methoxyethyl)(oxolan-3-ylmethyl)(thiophen-2-ylmethyl)amine
N-(1,3-benzoxazol-2-ylmethyl)-3-(3-hydroxy-3-methylbutyl)benzamide
{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
3,7-dimethyl-11-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}-3,7,11-triazaspiro[5.6]dodecane
1-[1-(3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-8-methylquinolin-2-yl)piperidin-4-yl]piperidin-4-ol
N-(1-{7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
1-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
methyl 8-(1-benzofuran-2-ylmethyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[1-methyl-4-(oxolan-3-ylmethyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]-2-phenoxyethan-1-one
[(4-fluorophenyl)methyl](methyl){[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[methyl({5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl})amino]ethan-1-ol