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2-(1-{1-[1-(4-fluorophenyl)piperidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(5-ethylfuran-2-yl)methyl]piperidine-4-carboxamide
3-(4-phenyl-1H-imidazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N3-[2-(cyclohex-1-en-1-yl)ethyl]-N5-(cyclopropylmethyl)-1-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
[1-(5-chloro-3-methyl-1H-indole-2-carbonyl)-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl]methanol
N-methyl-2-(5-methyl-3-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-1H-pyrazol-1-yl)acetamide
3-{[1-(1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
N-(2,3-dihydro-1H-inden-2-yl)-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-propylacetamide
N-[(5-chlorothiophen-2-yl)methyl]-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3R,4R)-1-(5-chloro-3-fluoropyridin-2-yl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
2-(propan-2-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,3-benzoxazole-5-carboxamide
1-(4-hydroxypiperidin-1-yl)-3-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
phenyl (7S,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
5-methyl-N-[2-(propan-2-yloxy)ethyl]-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(3R,4R)-1-(2,1,3-benzoxadiazole-5-carbonyl)-4-ethylpiperidine-3,4-diol
(3aS,6aS)-2-(2-chlorobenzoyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-(azocan-1-yl)-N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]propanamide
5-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(4aS,7aR)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,9aR)-1-[({3-[(pyridin-3-yl)amino]propyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
3-{[(2,5-dimethylphenyl)methyl]amino}-N-[3-(1H-imidazol-1-yl)propyl]-5-(pyrrolidine-1-sulfonyl)benzamide
2,5-dioxo-6-[2-(pyridin-3-yloxy)propyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-[(3-chlorophenyl)methyl]-5-cyclobutyl-1-methyl-1H-1,2,4-triazole
N-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
4-benzyl-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6-(morpholin-4-yl)pyrimidin-4-amine
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1-methylazepane-2-carboxamide
2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(3-methylbutyl)acetamide
1-(2-methylpropyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
N-(cyclopropylmethyl)-4-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]sulfamoyl}benzamide
N-(3-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-oxopropyl)acetamide
methyl 2-(2-{[3-(dimethylcarbamoyl)propanamido]methyl}-5-methyl-2,3-dihydro-1-benzofuran-7-yl)benzoate
3-methyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-oxo-2,3-dihydro-1,3-benzoxazole-5-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-(1-phenylcyclopropanecarbonyl)piperazin-2-yl}ethan-1-ol
4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-[(4-methylphenyl)methyl]pyridin-2-amine
2-(morpholin-4-ylmethyl)-4-(pyrimidin-5-yl)phenol
N-[1-(1-{[(4-chloro-3-methylphenyl)carbamoyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)ethyl]acetamide
2-(2-methyl-1,3-thiazol-4-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-3-carboxamide
2-[2-(3-fluorophenyl)ethyl]-4-{3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-[2-(4-fluorophenyl)ethyl]-5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
2-{[2-amino-6-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrimidin-4-yl]amino}ethan-1-ol
(1S,5R)-6-benzyl-3-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-cyclopentyl-3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-3-(3-fluorophenyl)pyrrolidine-2,5-dione
2-[1-(cyclohexylmethyl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-5-methoxy-1,4-dihydropyridin-4-one