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8-[2-(methylamino)pyridine-4-carbonyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(oxan-4-yl)pyridin-2-amine
11-{[(2-chlorophenyl)methyl]amino}-4-[(3-fluorophenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperazine
5-fluoro-4-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]quinazoline
8-methyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-2-(thiophen-2-yl)quinoline
methyl 6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-3-(5-methylthiophene-2-amido)thieno[2,3-b]pyridine-2-carboxylate
(1R,9S)-5-amino-3-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
2-[1-(1-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-amine
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-3-(1,2-oxazolidin-2-yl)propanamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)furan-3-carboxamide
4-methoxy-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
4-phenyl-3-(piperidin-3-yl)-1-[2-(propan-2-ylsulfanyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-[(3-methoxyphenyl)methyl]-4-[4-(methylsulfanyl)benzoyl]morpholine
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-(3-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-3-oxopropyl)pyrrolidin-2-one
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-4-(oxolan-2-ylmethyl)piperazine
6-[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
N-(2-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}propyl)acetamide
5-({2-[2-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)-2-(methylsulfanyl)pyrimidine
3-(pyrazin-2-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
methyl 3-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}pyrazine-2-carboxamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
4-[(4-{4-benzyl-5-[(pyridin-3-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-N,N-dimethylaniline
N,6-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]imidazo[1,2-a]pyridine-2-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]butan-1-one
({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)[1-(1H-pyrazol-1-yl)propan-2-yl]amine
6-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
N-[(1S,2R)-2-{[1-(2-chlorophenyl)piperidin-4-yl]amino}cyclobutyl]-2-(methylsulfanyl)acetamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-1-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
N-[3-(furan-2-yl)-3-phenylpropyl]-5-propyl-1,2-oxazole-3-carboxamide
ethyl 3-{2-[(2,5-dimethylphenyl)carbamoyl]acetamido}-4-methylpentanoate
4-methyl-N-[(1R,3S)-3-{[3-(4-methyl-1H-pyrazol-1-yl)propyl]carbamoyl}cyclopentyl]-1,3-oxazole-5-carboxamide
2-methyl-5-{1-[(3-methylphenyl)methyl]-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl}pyrazine
N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
1-[(5-methyl-4-phenyl-1H-imidazol-1-yl)methyl]cyclohexan-1-ol
1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
6-ethyl-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(piperidin-1-yl)pyrimidin-4-amine
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]oxane-2-carboxamide
(2S)-N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-4-methylpentanamide
({4-[1-(dimethylamino)ethyl]phenyl}methyl)({2-[(dimethylamino)methyl]phenyl}methyl)methylamine
1-({4-methyl-5-[1-(pyridin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(pyridin-4-yl)propanamide
8-(5-methyl-1,3,4-oxadiazol-2-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-hydroxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
dimethyl(2-{[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]oxy}hex-5-en-1-yl)amine